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6-(4,4-difluoropiperidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
4-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)morpholine
N-[(6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]acetamide
N-({7-[2-(2,5-dimethoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
2-[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]pyridine
[1-(3,5-dichloro-4-methylbenzoyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
3,5-dimethyl-1-({3-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-pyrazole
N-(2-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
(4aS,7aR)-1-(5-ethylthiophene-3-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(dimethyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2S,4S,6R)-2-(3-cyanophenyl)-6-(3,5-difluorophenyl)oxan-4-yl]acetamide
N-(3,4-difluorophenyl)-2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]acetamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(1H-imidazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(azepan-1-yl)-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{[3-(4-hydroxyphenyl)phenyl]methyl}acetamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}cycloheptanamine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methylpiperidine
N-benzyl-5-[(4-methoxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(3-fluorophenoxy)piperidin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
2-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}imidazo[1,2-a]pyrimidine
1-benzyl-3-(2-methylpropyl)-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-benzyl-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methyl}acetamide
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
[(3R,4S)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-methyl-6-[4-(thiophen-2-ylmethyl)piperazin-1-yl]pyrimidin-2-amine
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(1-phenylpiperidin-4-yl)piperidine-3-carboxamide
N3-[3-(dimethylamino)propyl]-1-[(2-methoxyphenyl)methyl]-N3-methyl-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidine-2-carboxylate
(2E)-3-(3-fluorophenyl)-N-{[3-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)prop-2-enamide
(3aR,6aR)-2-cyclopropanecarbonyl-N-[3-(morpholin-4-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-(3-hydroxy-2,2-dimethylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-[4-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
3-{[cyclopropyl(pyridin-2-ylmethyl)amino]methyl}-8-methyl-1,2-dihydroquinolin-2-one
4-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3-dihydro-1H-imidazol-2-one
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(thian-4-yl)piperidin-4-yl]imidazolidine-2,4-dione
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
2-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-[(2R,3R)-2-methoxy-1'-(1H-pyrazol-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
N-[(2,4-difluorophenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-[3-(benzenesulfonyl)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
ethyl 3-({2-[(1-acetylpiperidin-4-yl)oxy]-5-chlorophenyl}formamido)propanoate
2-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}-5-methoxyphenol
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
N-{4-[({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}carbamoyl)methoxy]phenyl}propanamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide