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N-[1-(furan-2-yl)ethyl]-N,2-dimethyl-3-[(pyridin-3-ylmethyl)amino]benzamide
4-(2-methylpropyl)-3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
N-[(2R,3R)-1'-(3-fluoro-4-methoxybenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1-methylazepane-2-carboxamide
N-{4-[2,2-bis(hydroxymethyl)butanamido]phenyl}-4-methylbenzamide
2-(4-{[(3S,4S)-3,4-dihydroxypiperidin-1-yl]methyl}phenoxy)acetic acid
N-(1-methanesulfonylpiperidin-4-yl)-2-[(prop-2-en-1-yl)amino]benzamide
(2S,4S)-4-amino-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-N-ethylpyrrolidine-2-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
3-ethoxy-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
(1S)-1-[1-benzyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine
N-cyclopropyl-3-{1-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]piperidin-3-yl}propanamide
methyl 3-({[1-(pyridin-2-ylmethyl)piperidin-4-yl]carbamoyl}amino)benzoate
5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-(2-phenylpropyl)-1H-pyrazole-4-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-3-(pyrrolidine-1-carbonyl)-1,2-oxazole
N-[2-(3-fluoro-4-methylphenyl)phenyl]cyclopropanecarboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2,2-dimethylpropanoyl)piperidine-2-carboxamide
1-[2-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-amino-3-ethyl-N-methyl-N-(quinolin-5-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-phenyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-methoxy-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N,N-dimethyl-2-[(3-methyl-2-phenylbutanamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-(3-methylphenyl)-3-[2-(phenylamino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(cyclopentylmethyl)-N-[2-(diethylamino)ethyl]-1-(2-methoxyethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-benzyl-9-(4-methoxypyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-{1-[1-(1-ethyl-3-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-[(2R)-2-amino-2-cyclohexylacetamido]-N-(3-methoxyphenyl)benzamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]piperidine-3-carboxamide
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-methylbutanamide
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-methyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]cyclohexane-1-carboxamide
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}isoquinoline
1-cyclopentanecarbonyl-3-(4-methoxyphenoxymethyl)piperidine
N-[(3S,4R)-1-[2-(3,4-dimethylphenoxy)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-cyclopropanecarbonyl-8-[4-(dimethylamino)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[7-acetyl-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-N-ethylpyrrolidine-3-carboxamide
6-(3-chlorophenyl)-2-(4-hydroxypiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-N,1-dimethylpiperidin-4-amine
3-(2-ethyl-1H-imidazol-1-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyridin-2-amine
2-(3-phenylpropyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1,3-benzoxazole
9-(1H-imidazole-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}azetidin-3-ol
N-[1-methyl-2-phenyl-7-(pyrrolidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]ethane-1-sulfonamide
2-(pyrimidin-5-yl)quinoxaline
6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5S,8R)-8-methoxy-3-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-azabicyclo[3.2.1]octane