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{[2-methoxy-5-(4-phenyl-1H-imidazol-5-yl)phenyl]methyl}dimethylamine
1-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-{3-[(3,4-dimethoxyphenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}ethyl)pyrazine
2-(adamantan-1-ylsulfanyl)-1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)ethan-1-one
N-butyl-N-[(2-fluorophenyl)methyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
2-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1,3-benzothiazole
5-{[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
N4-[(2,6-difluoro-3-methoxyphenyl)methyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
2-(3-chlorophenyl)-1-[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
(4aR,8aS)-1-(cyclohexylmethyl)-6-(naphthalen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(3-methoxyphenoxy)-N-[(1-methylpiperidin-3-yl)methyl]acetamide
N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}oxan-4-amine
4-hydroxy-2-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)quinoline-6-carboxamide
(1R,5R)-N-(5-chloro-2-methylphenyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N5-butyl-N2-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2,5-dicarboxamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-3-(piperidin-3-yl)benzamide
N-{[1-(4-cyanopyridin-2-yl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
3-methyl-1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-3-phenylpiperidine
2-(4-fluorophenyl)-N-[2-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
ethyl 4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidine-1-carboxylate
2,2-dimethyl-N-(3-{[3-(6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-1-yl]methyl}pyridin-2-yl)propanamide
3-ethyl-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
N3-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-{2-[2-(methylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-1-phenylcyclopropane-1-carboxamide
2-[({[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}amino)methyl]-3,4-dihydroquinazolin-4-one
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]ethan-1-one
8-(2-ethylpyrimidine-5-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N,1-dimethyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(3S,4R)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
(1R,5R)-N,N-dimethyl-6-[2-(pyridin-2-ylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-cyclopropyl-9-(cyclopropylmethyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
N-(1,4-dioxan-2-ylmethyl)-4-(piperidin-1-ylmethyl)benzamide
6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-9H-purin-2-amine
4-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-ethylpyrrolidin-2-one
2-[methyl({[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1-phenylethan-1-ol
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
9-(4-methoxy-2,3,6-trimethylbenzenesulfonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
8-{2-[methyl(propan-2-yl)amino]acetyl}-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(3-methoxypropyl)-9-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-(pyrrolidin-1-yl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-[2-(1H-indol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(1-methyl-5-oxopyrrolidin-2-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(1H-1,3-benzodiazol-1-yl)-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidine-4-carboxylic acid
2-(1-cyclohexylpyrrolidin-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-benzyl-1-methyl-5-(quinoxaline-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
4-(1-hydroxy-2-phenylethyl)-N-(quinolin-7-yl)piperidine-1-carboxamide