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N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(thiophen-3-yl)acetamide
(1R,5R)-3-(3-chlorobenzoyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
1-[3-({[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]amino}methyl)pyridin-2-yl]piperidin-3-ol
1-(3-chlorophenyl)-3-(2-methoxyethyl)-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazole
1-({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)-4-methylpiperidine-4-carbonitrile
N-[3-(1H-imidazol-1-yl)propyl]-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[4-(difluoromethoxy)phenyl]-2-propylpyrrolidine-1-carboxamide
4-{[3-(2-{4-[4-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}morpholine
N-(4-{[3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
(3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl)methanol
(1-methyl-1H-imidazol-2-yl)(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)methanol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-[(2-methoxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
3-(pyrrolidine-1-carbonyl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}benzene-1-sulfonamide
2-(2-chloro-6-fluorobenzamido)-N-[2-(2-fluorophenyl)ethyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]methanol
1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
3-methoxy-N-(1-{7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2,4-dimethyl-N-{4-[4-({[1-(propan-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]phenyl}benzamide
3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-1-[3-(trifluoromethoxy)phenyl]urea
1-(4,4-difluoropiperidin-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
5-{2-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
9-methoxy-3-(3-phenyl-1,2-oxazole-5-carbonyl)-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-cyclopropyl-2-[(2-methylprop-2-en-1-yl)oxy]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,2-dimethyl-1H-1,3-benzodiazole-5-carboxamide
(1S,4S)-2-(3-chlorophenyl)-5-[2-(2-methyl-1H-indol-3-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
ethyl 4-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}piperidine-1-carboxylate
1-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-[(3,4-dimethylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
1-[1-(3-methylbenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-[(2R)-2-amino-3-methylbutanoyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-({[2-(1H-indol-1-yl)ethyl]amino}methyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
1-{3-[3-(pyridin-4-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
2-methyl-4-phenyl-9-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-methyl-N-(2-phenyl-1-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl)-2-(1H-pyrazol-1-yl)acetamide
(3R,4S)-1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3,4-dimethylpiperidin-4-ol
(4aR,8aS)-6-[(2,4-dimethylphenyl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
2-(2,4-difluorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
6-[6-oxo-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
1-(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-N-(propan-2-yl)piperidine-4-carboxamide
1-{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}-2,5-dihydro-1H-pyrrole
N-methyl-N-{2-phenyl-1-[1-(quinolin-5-ylmethyl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
methyl 1-[2-hydroxy-3-(3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)propyl]piperidine-4-carboxylate
1-(cyclohexylmethyl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-6-oxopiperidine-3-carboxamide