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6-chloro-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyridazin-3-amine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4-sulfamoylbenzamide
1-[7-(oxolane-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-4-ol
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine
5-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(2-methylpyridin-4-yl)methyl]piperidine-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-3-phenyl-1H-pyrazole-5-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-methoxy-6-methyl-4-(3-methylthiophen-2-yl)-1,2,3,4-tetrahydroquinolin-2-one
[(3S,7S)-5-(thiophene-2-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methoxyacetamide
2-[3-(pyridin-2-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(2-oxocyclopentyl)acetamide
2-(3-methoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[3-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-1-yl)propyl]amine
1-cyclohexyl-N3-(2-methylpropyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]pyrrolidin-2-one
N-({1-[(2-ethylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N,N-dimethyl-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)but-3-enamide
N-[3-(4-chlorophenyl)propyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]acetamide
3-[5-(1H-indol-2-yl)-1,3,4-oxadiazol-2-yl]-N-(1-methoxybutan-2-yl)propanamide
2-ethyl-N-[1-(pyrimidin-4-yl)ethyl]pyrimidine-5-carboxamide
3-[2-(dimethylamino)ethyl]-8-(5-propyl-1,2-oxazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3,4-dimethoxyphenyl)-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{spiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
1-(3-{[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)amino]methyl}phenyl)ethan-1-one
N-(6-chloropyridin-3-yl)-4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carboxamide
3-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3,4-dihydro-2H-1,4-benzoxazine-6-sulfonamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
4-({3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-oxobutanamide
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-(3-phenylpropyl)piperidin-2-one
2-{5-[1-(1H-pyrazol-1-yl)propyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-N,N-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-(oxolan-2-ylmethyl)propanamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{4-[4-(piperazin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(hydroxymethyl)-2-methyl-4-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}pyridin-3-ol
dimethyl({4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]phenyl}methyl)amine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidin-3-yl]methanol
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-hydroxyethyl)acetamide