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ethyl 4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazine-1-carboxylate
2-[2-(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
5-[2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
2-{5-[(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}pyridine
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-4-(1H-imidazol-1-yl)-N-(pyridin-4-ylmethyl)benzamide
(2E)-N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
2-[4-(1,3-oxazol-5-yl)benzoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(3-methylbutyl)-5-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-(3,6-dimethylpyrazin-2-yl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(propane-2-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-{7-[(2-chloro-6-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
1-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-4-(2-methoxyethyl)piperazine
2-[(3-methoxyphenyl)methyl]-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}morpholine
(3S,4R)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-methoxypiperidin-4-amine
1-[2-(azepan-1-yl)-2-oxoethyl]-4-benzyl-3-butyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
4'-(2-phenylethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-(2,2-dimethylpropyl)-2-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,7-diazaspiro[4.5]decane
5-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-1,2-oxazole-3-carboxamide
3-[(cyclobutylamino)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-methyl-2-(5-methylfuran-2-yl)-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-5-(1H-imidazol-1-ylmethyl)furan-2-carboxamide
N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylbut-2-enamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(4-fluorophenyl)piperazine
2-[4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
5-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}-N-methylfuran-2-carboxamide
3-(2-amino-4-{[(5-methoxy-1H-indol-2-yl)methyl]amino}-6-methylpyrimidin-5-yl)propanoic acid
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
3-cyclopentyl-1-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
N-[cyclopropyl(4-methoxyphenyl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
4-{1-[(3-fluoropyridin-4-yl)methyl]piperidin-4-yl}thiomorpholine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
2-ethoxy-3-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-(methylsulfanyl)-N-[2-(piperidin-1-yl)ethyl]acetamide
(4aR,8aR)-7-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
N-{2-[1-(4-propylphenyl)-1H-imidazol-4-yl]ethyl}acetamide
3-{1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}phenol
3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}-N-(1,3-thiazol-2-yl)propanamide
4-methoxy-N-{1-[1-(3-phenylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
methyl(2-phenylethyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-[(2-chloro-5-fluorophenyl)methyl]azepan-2-one
(4S)-3-{2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-methoxypyrimidin-4-amine
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}isoquinoline
methyl 3-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzoate
2,3-dimethyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}quinoxaline-6-carboxamide
6-(3-chloro-4-fluorobenzoyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(3-hydroxyphenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-(4-fluorophenyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)-1,2,3,6-tetrahydropyridine
3-methyl-8-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one