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ethyl 1-(4-fluorophenyl)-5-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-4-carboxylate
N-[(2-chloropyridin-3-yl)methyl]-2-(2,3-dihydro-1H-inden-1-yl)-N-methylacetamide
4-benzyl-3-ethyl-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,4-diazepan-5-one
6-methyl-3-{1H-pyrazolo[3,4-b]pyridin-1-yl}pyridin-2-amine
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-2-[2-(methoxymethyl)piperidin-1-yl]pyridine
2-({4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}methyl)pyridine
N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
2-(ethylamino)-N-[2-(propan-2-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenoxy)-N-(propan-2-yl)piperidine-4-carboxamide
1-(2-fluorobenzoyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-methoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
(1R,5R)-6-benzyl-3-(1-phenyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 1-(cyclohexylcarbamoyl)-4-(2-phenylethyl)piperidine-4-carboxylate
2-(3-fluorophenyl)-N-({7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
N-(3,4-dimethylphenyl)-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
9-(5-chloro-2-hydroxybenzoyl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methoxyphenyl)-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
1-{2-[(4-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N,N-bis(prop-2-en-1-yl)piperidine-4-carboxamide
N-[(1-ethylpiperidin-3-yl)methyl]-7-methoxy-N,4-dimethylquinazolin-2-amine
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-indole-6-carboxamide
2-fluoro-N-(1-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)benzamide
N-benzyl-N-butyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
methyl[2-(1H-pyrazol-1-yl)ethyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}-N-cyclopropylpropanamide
9-(1-ethyl-1H-pyrazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
methyl(naphthalen-1-ylmethyl)[(4-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(4-chlorophenyl)methyl]amino}piperidin-1-yl)benzamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1H-1,2,3-benzotriazol-1-yl)propan-1-one
5-[(4-chlorophenyl)methyl]-5-{3-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-chloro-N-cyclopropyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}benzamide
7-methoxy-1-methyl-2-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
(2R,3R)-3-amino-1'-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
3-cyclobutyl-N-(4-methyl-2-oxo-2H-chromen-7-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
1-[1'-(2-methoxy-5-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-{[3-(2-methylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
(1H-imidazol-2-ylmethyl)[(3-{[1-(4-methoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl]methylamine
5-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
(1R,5R)-N,N-dimethyl-6-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-ol
2-{1-[(2-fluorophenyl)methyl]-4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-2-yl}ethan-1-ol
4-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
4-methoxy-N-[(3-methylphenyl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
3-(5-methylfuran-2-yl)-N-{3-[(pyridin-3-yl)amino]propyl}-1H-pyrazole-5-carboxamide
2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
(cyclohexylmethyl)({[2-(4-ethylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl})amine
2-(5-methyl-1,2-oxazol-3-yl)-1-(2-phenylethyl)piperidine