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N-cyclohexyl-4,5,6-trimethyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-(3-cyclopentylpropyl)-1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
methyl 4-(5-chloro-2-{[2-(2-methyl-1,3-thiazol-4-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
N-(3,4-dimethoxyphenyl)-1-[3-(trifluoromethyl)benzoyl]piperidin-3-amine
(3S,4S)-1-[3-(morpholin-4-yl)benzoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-butyl-1'-(3-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3R,4R)-1-(5,6-dimethylpyrimidin-4-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-7-methoxy-4-methylquinazoline
5-ethyl-3-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
4-[(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}furan-2-yl)methyl]morpholine
1-(4-methoxyphenyl)-5-(5-methyl-1,2-oxazol-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
N-[2-(4-methoxyphenyl)phenyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2H-1,3-benzodioxol-5-yloxy)acetamide
3-ethyl-1-[(8-methoxyquinolin-2-yl)methyl]piperidine-3-carboxylic acid
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-4,4,4-trifluorobutan-1-one
N-(1-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)azepan-4-amine
2-(methylamino)-N-(prop-2-en-1-yl)-N-(propan-2-yl)benzamide
3-{5-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}benzonitrile
1-[5-(2-chloro-4-fluorobenzoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-ethyl-5-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}pyrimidin-2-amine
N,N-diethyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamide
(3R,4S)-4-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
3-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,5-dimethylpyrazine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]ethan-1-one
(4aS,8aR)-6-(3-cyclopropylpropanoyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
3-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-N-(propan-2-yl)propanamide
6-(2-methoxyphenyl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(3,5-dimethoxyphenyl)methyl]({[8-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl})amine
N-{1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylpyrimidin-2-amine
1-{2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]ethyl}-2,3-dihydro-1H-imidazol-2-one
N-cyclohexyl-3-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}formamido)propanamide
2-{[(2,2-dimethyloxan-4-yl)(ethyl)amino]methyl}benzonitrile
4-(5-methoxyfuran-2-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-(3-fluorophenoxy)-1-(3-fluoropyridin-4-yl)piperidine-4-carboxylic acid
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-7-fluoro-2-methylquinoline-4-carboxamide
N-benzyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-(oxolan-2-ylmethyl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-(2-methoxyphenyl)-4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidine
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(3-fluorophenoxymethyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,3-oxazole-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]ethan-1-one
8-[(4-fluoro-3-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-butyl-2-methyl-N-[(3-methylthiophen-2-yl)methyl]-3-(1H-pyrazol-1-yl)propanamide