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2-(1-ethyl-3-oxopiperazin-2-yl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
8-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-5-(2-methylbutanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
2-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(1-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-({7-[(2E)-3-(4-chlorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N,N,2-trimethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(oxolane-2-carbonyl)-4-[4-(pyrrolidin-1-ylmethyl)phenoxy]piperidine
1-(4-methoxyphenyl)-4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidine
[(1-ethyl-1H-imidazol-5-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
N-(2-{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]morpholin-2-yl}ethyl)-2,2-dimethylpropanamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinolin-4-yl)piperidin-3-yl]propanoic acid
{9-[(4-fluorophenyl)methyl]-3-(1,2-oxazole-3-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
2-(cyclopent-1-ene-1-carbonyl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
N-{2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-1-methylpiperidine-3-carboxamide
methyl (2S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[2-chloro-5-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
2-phenyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
3-methyl-N-{1-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
3-(2-methoxyethyl)-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
2-ethyl-1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-2,5-dihydro-1H-pyrrole
6-[3-(4-methylphenyl)propanoyl]-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(1R,5S,6S)-6-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-methylpiperidin-2-one
1-(oxan-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[benzyl(methyl)amino]-3-[5-({[3-(dimethylamino)propyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-[(3R,4R)-3-hydroxy-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl]pyrazine-2-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-(furan-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-methyl-3-propyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}-1H-pyrazole-5-carboxamide
1-[(3R)-3-cyclopropyl-3-hydroxy-4,4-dimethylpyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
3-benzyl-3-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-1-methyl-2,3-dihydro-1H-indol-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2-hydroxybutyl)-1,3-oxazole-4-carboxamide
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidine
methyl 1-{[4-(5-methoxy-5-oxopentanoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-2-carboxylate
2-(furan-2-yl)-2-oxo-N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
(1R,5R)-6-(cyclobutylmethyl)-3-(2,6-difluoro-4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethylpiperidine-2-carboxamide
3-chloro-6-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-2-carboxylic acid
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-[(3S)-2-oxoazepan-3-yl]piperidine-3-carboxamide
2-(2-aminoacetyl)-N-(cyclopropylmethyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-1,3-dimethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-5-carboxamide
3-(2-methoxyethyl)-3-methyl-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea