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N-({7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)propane-2-sulfonamide
[(3R,4R)-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-({3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-2,6-dimethoxyphenol
(2S,4R)-4-amino-1-[4-(difluoromethoxy)benzenesulfonyl]-N-methylpyrrolidine-2-carboxamide
N-{2-[1-butyl-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-(dicyclopropylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-ethyl-4-[3-(4-fluorophenoxy)azetidin-1-yl]-6-methylpyrimidin-2-amine
N,N-dimethyl-4-[4-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-4-oxobutanamide
6-methyl-4-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-[(3-chlorophenyl)methyl]-N-ethyl-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-cyclopropyl-5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}piperidin-2-one
9-methoxy-3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(5-fluoro-2-methylphenyl)methyl]benzamide
(3S,9aR)-3-(cyclohexylmethyl)-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-3-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3-methylpyridin-2-yl)methyl]piperidine-3-carboxamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-acetyl-8-[3-(4-hydroxyphenyl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(1,3-dihydroxypropan-2-yl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
9-(6-aminopyridine-3-carbonyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
6-chloro-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}imidazo[2,1-b][1,3]thiazole
1-benzyl-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-1H-pyrazole-4-carboxamide
3-chloro-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-butyl-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
2-(5-ethylfuran-2-yl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
2-amino-4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-(2-methoxyethyl)-5-{[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}pyrimidine
5-(oxolan-2-yl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]thiophene-2-carboxamide
{7-fluoro-5-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
4-(2,6-dimethylpyrimidine-4-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
4-(4-chlorophenoxy)-1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-methyl-N-(oxan-4-ylmethyl)-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-(3,4-dimethoxyphenyl)-1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
methyl 7-oxo-3-(3-phenylpropanoyl)-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-cyclopropyl-3-{1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(6-methylpyridin-2-yl)ethyl]acetamide
2-[(4-chlorophenyl)methyl]-5-(4-methoxypiperidine-1-carbonyl)-1,3-benzoxazole
2-methyl-1-(3-{2-[2-(morpholin-4-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}piperidin-1-yl)propan-1-one
2-ethyl-5-{[3-(3-methylphenyl)piperidin-1-yl]methyl}pyrimidine
1-methyl-5-[4-(propan-2-yloxy)phenyl]-1H-imidazole
N-(adamantan-2-yl)-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(2-hydroxyethyl)-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-[2-(4-phenylpiperidin-1-yl)ethyl]-1,3-benzothiazole-6-carboxamide
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-7-oxo-N-(2-phenylethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)butan-1-one
4-{6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carbonyl}morpholine
1-(2-{[6-(2-methoxyphenyl)pyridazin-3-yl]amino}ethyl)imidazolidin-2-one
[3-(furan-2-ylmethyl)-9-(3-methoxypropyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol