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1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(3,5-difluorobenzoyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
4-(5-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
3-methyl-1-(2-methylpropyl)-4-(5-phenylpentanoyl)piperazin-2-one
2-[(dimethylamino)methyl]-N-[3-(1H-indol-1-yl)propyl]-1,3-thiazole-4-carboxamide
8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidin-4-ol
ethyl 4-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}butanoate
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
2-(hydroxymethyl)-N-[2-(trifluoromethoxy)phenyl]piperidine-1-carboxamide
4-(2,3-dimethoxyphenyl)pyrimidine
2-cyclopentyl-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-[(1-phenylcyclohexyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
2-ethyl-5-{1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidine
1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-(1H-indol-5-yl)-4-(morpholin-4-yl)piperidine-1-carboxamide
4-{2-[(6-cyclopropylpyrimidin-4-yl)amino]-1-hydroxyethyl}phenol
3-(3-hydroxy-1,2-oxazol-5-yl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)propan-1-one
2-[(7-chloro-2-methylquinolin-4-yl)formamido]-N,N,3-trimethylbutanamide
1-[2-methoxy-4-({[2-(naphthalen-1-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-4-methyl-2-phenylpyrimidine-5-carboxamide
2-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyridine
(2S,4R)-N-ethyl-4-(3-hydroxypropanamido)-1-[(1-methyl-1H-indol-6-yl)methyl]pyrrolidine-2-carboxamide
2-methoxy-2-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
2-methoxy-1-[1'-(4-methylpyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
2,2-dimethyl-1-{2-[5-(morpholine-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}propan-1-one
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
2-methoxy-1-[4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,4-diazepan-1-yl]ethan-1-one
4-(3-ethoxypropanoyl)-1-phenylpiperazin-2-one
(2S,4S)-N-ethyl-4-[2-(methylsulfanyl)acetamido]-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
2-(2-acetyl-1H-1,3-benzodiazol-1-yl)-N-(1-methyl-1H-indazol-3-yl)acetamide
methyl 3-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(ethylamino)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}pyrimidine-5-carboxamide
6-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
4-[(2-fluorophenyl)methyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
3-methyl-1-{1-[6-(pyrrolidin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
N-(3,4-dimethoxyphenyl)-3-[(2-methylpyrrolidin-1-yl)methyl]benzamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylbenzamide
N-cyclopropyl-1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidine
1-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-fluoro-N,5-dimethylimidazo[1,2-a]pyridine-2-carboxamide
7-(4-methoxybenzoyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
[2-(2-chloro-6-fluorophenyl)ethyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-methyl-3-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,4-dihydroquinolin-4-one