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N-[(1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
1-benzyl-N,N-dimethyl-5-{[(2-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(1-methylpiperidin-2-yl)-N-[2-(pyridin-4-yl)ethyl]propanamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-[(3R,4S)-4-(dimethylamino)-1-[(2-fluoro-5-methylphenyl)methyl]piperidin-3-yl]propan-1-ol
N-ethyl-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]pyrimidin-2-amine
3-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[2-(morpholin-4-yl)ethyl]urea
3-(4-methyl-1,3-thiazol-5-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
1-[2-(4-phenylphenyl)acetyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
3-({4-[1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
2-(1H-imidazol-2-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]benzamide
2-cyclopropyl-6-oxo-N-(propan-2-yl)-N-(2,2,2-trifluoroethyl)-1,6-dihydropyrimidine-5-carboxamide
N-[2-(morpholin-4-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-(1-benzoylpiperidin-3-yl)pyrimidin-2-amine
2-{4-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
6-{[benzyl(ethyl)amino]methyl}-2-oxo-N-[1-(thiophen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
4-[(2-chlorophenyl)methyl]-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3-methylbutyl)-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[4-(isoquinolin-5-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
4-(1H-imidazol-1-yl)-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}benzamide
(1-methanesulfonylpropan-2-yl)({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl})amine
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-{[7-(4-carbamoylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-methoxyethyl)acetamide
1-(2-phenylethyl)-N-[(3-phenylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
ethyl 2-(1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazol-4-yl}-N-methylformamido)acetate
N-cyclopentyl-1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
4,5-dimethyl 1-[(3S,5S)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N2-cyclopropyl-N4-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-{2-[3-(4-fluoro-2-methoxyphenyl)phenoxy]ethyl}-1H-imidazole
2-[(3,4-dimethoxyphenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-N,N-dimethylpyrrolidin-3-amine
(1R,5S,6R)-3-(2,1,3-benzoxadiazol-4-ylmethyl)-N-(pyridin-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-(1-{1-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-2-phenylethyl)-N,2-dimethylpropanamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[4-(1H-pyrazol-3-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-3-enamide
1-(2,4-difluorobenzoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
3-(3-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzoic acid
2-[benzyl(methyl)amino]-N-[(2S)-pyrrolidin-2-ylmethyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl 1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
2-ethyl-5-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
methyl 1-[(3R,5S)-1-(2-methylpropyl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
6-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]pyridine-2-carboxylic acid
7-cyclohexyl-2-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one