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N-[(5-methylpyrazin-2-yl)methyl]-1-(quinoxalin-2-yl)piperidin-4-amine
8-[(1-acetyl-1H-indol-3-yl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-(dimethylamino)ethyl]-9-(furan-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxane-2-carboxamide
N-methyl-3-(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)-N-(1-methylpiperidin-4-yl)propanamide
3-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-N-(pyridin-3-yl)benzamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
N-[(3S,4R)-1-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-{[3-(methylsulfanyl)phenyl]methyl}-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
2-methoxy-2-phenyl-1-(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-methyl-5-{[3-(4-methyl-3-phenylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-1,3-benzothiazole
2-[(4-methylphenyl)methyl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
1-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-6-(cyclobutylmethyl)-3-[(2-cyclohexylpyrimidin-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(6-ethoxyquinolin-2-yl)methyl]-N-methylpiperidine-2-carboxamide
1-[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazol-3-yl]ethan-1-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
N-(pyridin-3-ylmethyl)-4-(quinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-{1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
2-ethyl-5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyrimidine
1-(2-methoxyphenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
6-[(3,4-dimethoxyphenyl)methyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
5-(adamantane-1-carbonyl)-1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 1-(1H-indazol-6-yl)-1H-imidazole-2-carboxylate
8-cyclopropanecarbonyl-2-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methoxy-6-(propan-2-yl)-3-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(2-oxo-2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-3-methylthiophene-2-carboxamide
{2-[(4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)methyl]phenyl}methanol
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-fluorophenyl)-1,4-diazepane
3-(4-methylpiperazine-1-carbonyl)-N-[(1-phenylcyclohexyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3,5-dimethyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-benzofuran-2-carboxamide
5-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-2-amine
5-(4-methoxyphenyl)-N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,2,4-triazin-3-amine
1-[3-oxo-3-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)propyl]pyrrolidin-2-one
N-(4-methoxy-3-pentanamidophenyl)-3,5-dimethyl-1H-pyrrole-2-carboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
4-fluoro-N-{3-oxo-3-[3-(propoxymethyl)pyrrolidin-1-yl]propyl}benzamide
(1S,5R)-6-[4-(1H-pyrazol-3-yl)benzoyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-3,4-dihydropyrimidin-4-one
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-4-hydroxy-1-methylpiperidine-4-carboxamide
4-chloro-3-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
4-(1-hydroxy-2-phenylethyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-butyl-3-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidine
(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-2-yl)methanol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-3-({methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzamide