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N-(2-methoxyethyl)-4-[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)amino]pyridine-2-carboxamide
N-[2-(2-chlorophenyl)ethyl]-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[4-(trifluoromethyl)phenyl]ethyl}acetamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(2-phenoxyethyl)piperazine
3-{[(2-cyclooctylethyl)amino]methyl}-3-hydroxy-1-methylpiperidin-2-one
N-{[(3S,4S)-3-hydroxy-1-[2-(propan-2-ylsulfanyl)acetyl]piperidin-4-yl]methyl}morpholine-4-carboxamide
2-(1H-imidazol-1-yl)-N-{[3-methyl-7-(4-phenylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}acetamide
3-{[(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)amino]methyl}pyrrolidin-3-ol
methyl({[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl})(quinoxalin-6-ylmethyl)amine
3-benzoyl-1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidine
5,5-dimethyl-1-{2-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,6-dimethylphenol
3-{[(2-ethylphenyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
N-[(1R,3R)-3-aminocyclopentyl]-2-hydroxy-5-(morpholine-4-sulfonyl)benzamide
1-(2,3-dimethylphenyl)-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperazine
4-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,2-dimethylpiperazine
methyl 2-({4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}methyl)-1,3-oxazole-4-carboxylate
2-{[(3R,4S)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]methyl}benzoic acid
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-8-methylimidazo[1,2-a]pyridine-2-carboxamide
(2S,4S)-4-amino-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3-(2-phenylethyl)piperidine-3-carboxylate
N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
4-ethyl-3-{1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(furan-2-ylmethyl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]piperidine-4-carboxamide
1'-[3-(1H-1,2,4-triazol-1-yl)propyl]spiro[indene-1,4'-piperidine]
2-(3-methylpentanamido)-7-oxo-N-[(4-phenyloxan-4-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
7-[(4-fluorophenyl)methyl]-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(cyclopropylmethyl)-4-{[(2-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-methyl-8-[3-(1H-pyrazol-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
2-{3-methyl-5-[4-(1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl}pyridine
2-methyl-5-(3-methylphenyl)-4-[1-(oxolane-3-carbonyl)piperidin-3-yl]pyrimidine
1-ethyl-3-methyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
3-methyl-6-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}pyridazine
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
1-[(5-methylfuran-2-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
5-{3-[4-(1,3-benzoxazol-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-5-[(4-methoxyphenyl)methyl]pyrrolidin-2-one
(2R,6R)-11-methoxy-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyridazine
1-(4-methoxyphenyl)-4-[1-(3-methylbenzenesulfonyl)piperidin-3-yl]piperazine
ethyl({[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
7-[(2,3-difluorophenyl)methyl]-2-(1-propylpiperidin-4-yl)-2,7-diazaspiro[4.5]decane
methyl (2S)-1-[(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]pyrrolidine-2-carboxylate
4-{2-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
1-ethyl-2-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
methyl(1H-pyrazol-3-ylmethyl){[2-(trifluoromethoxy)phenyl]methyl}amine
(3R,4S)-4-[ethyl({[4-(3-hydroxy-3-methylbutyl)phenyl]methyl})amino]oxolan-3-ol
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine