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N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-[2-(3-chlorophenyl)ethyl]-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
1-[(3-hydroxyphenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
5-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
3-{[(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
(3aR,6aR)-2-cyclopentanecarbonyl-5-(3,5-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
N-[(1-methylpiperidin-4-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-[5-(1H-indol-6-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
2-ethyl-3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,2,3,4-tetrahydroisoquinoline
(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
N-methyl-2-(3-{[methyl({2-[4-(propan-2-yl)phenoxy]ethyl})carbamoyl]amino}phenyl)acetamide
(3S,9aR)-8-[(5-chlorothiophen-2-yl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-[(4-methylphenyl)sulfanyl]propan-1-one
4-[(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-1H-pyrazole-3-carboxylic acid
4-(propan-2-yl)-6-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]-2-(trifluoromethyl)pyrimidine
(5S,9aS,9bS)-2-methyl-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-(2-chlorophenyl)-2-[(3R)-3-methylpiperazine-1-carbonyl]-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(propane-1-sulfonyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(azocan-1-yl)propanamide
(1S,5R)-3-(3,4-difluorobenzoyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-1,4-diazepan-5-one
3-(2-chlorophenyl)-3-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)pyrrolidine-2,5-dione
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
4-hydroxy-N-[(2-methoxyphenyl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
8-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-benzyl-3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-2,8-diazaspiro[4.5]decane
1-(4-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
2-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
2-{1-[3-(methylsulfanyl)propyl]azetidin-3-yl}-1H-1,3-benzodiazole
3-[2-(furan-2-yl)azepane-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
(3aR,5R,6S,7aS)-2-(1H-1,2,3-benzotriazole-5-carbonyl)-octahydro-1H-isoindole-5,6-diol
1-[3-({2-[1-(2-methoxyethyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)piperidin-1-yl]ethan-1-one
2-{2-[2-(2,3-difluorophenyl)-1H-imidazol-1-yl]ethyl}piperidine
3-chloro-N-(4-pentanamidophenyl)pyridine-4-carboxamide
N-(cyclopropylmethyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[1-({1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
9-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-[(3-fluorophenyl)methyl]-6-methyl-3-(3-methylpiperidine-1-carbonyl)-1-[3-(morpholin-4-yl)propyl]-1,4-dihydropyridin-4-one
8-acetyl-2-[(2-aminopyridin-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-{[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(naphthalen-1-ylmethyl)piperazin-2-yl}ethan-1-ol
1-ethyl-8-(furan-3-ylmethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(4-fluorophenyl)-2-[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylacetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N,5,6-tetramethylpyrimidin-2-amine