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N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methylbenzamide
4-[(3-fluorophenyl)methyl]-1-[2-(1H-indol-3-yl)acetyl]-1,4-diazepan-5-one
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]pyridine-3-carbonitrile
N-[(2-chlorophenyl)methyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyloxane-2-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(3-hydroxypiperidin-1-yl)acetamide
N-[(2R)-1-oxo-1-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]propan-2-yl]acetamide
2-({[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]pyridine-2-carboxylic acid
5-[(3-methoxyphenyl)methyl]-3-methyl-5-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{4-[4-({[3-(trifluoromethoxy)phenyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-ol
4-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
5-{[5-(2,5-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1-methylpyrrolidin-2-one
N-cyclooctyl-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-{[4-(diethylamino)phenyl]methyl}-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-[1-(propan-2-yl)cyclopropyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(furan-2-yl)propan-1-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-methylthiophen-2-yl)methyl]amino}pyrrolidine-2-carboxamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-4-(thiophen-2-yl)butan-1-one
(3S,4S)-4-methyl-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperidine-3,4-diol
3-{[ethyl(methyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
N-(3-fluorophenyl)-4-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-4-oxobutanamide
5-cyclopropyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1,2-oxazole-3-carboxamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
2-methyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(3-fluorophenyl)-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyridine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
ethyl[(4-methanesulfonylphenyl)methyl][(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
(2E)-3-(4-methoxyphenyl)-1-{3-[5-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
9-methoxy-3-[(4-methoxyphenyl)methyl]-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(3-methoxypropyl)-1-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperidine-3-carboxylic acid
2-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
methyl 3-acetamido-5-[(2-ethylbutyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 4,4,4-trifluoro-3-{2-[(4-methylphenyl)carbamoyl]acetamido}butanoate
ethyl 4-[(4-chlorophenyl)methyl]-1-(3-ethynylbenzoyl)piperidine-4-carboxylate
6-methyl-2-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}methyl)quinolin-4-ol
N-[4-(2-fluorophenoxy)phenyl]-1-(oxane-2-carbonyl)piperidine-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-(1,2-oxazinan-2-yl)propanamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
5-(1-benzofuran-2-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,2,4-triazin-3-amine
5-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}pentan-1-ol
6-(3-methoxyphenyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(methylsulfanyl)propan-1-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[(3-methylthiophen-2-yl)sulfonyl]piperidine
3-benzyl-4-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
(1R,5R)-6-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-methyl-1H-1,3-benzodiazole-5-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[3-(methylsulfanyl)propyl]piperidine-3-carboxamide
(3S,4R)-1-[2-oxo-2-(piperidin-1-yl)ethyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-(1H-imidazol-1-yl)-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid