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4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-methyl-1,2,4-oxadiazole
1-(3,5-difluorophenyl)-N-[(3-ethoxy-4-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}pyridine
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(naphthalen-2-yl)ethan-1-one
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethylfuran-2-carboxamide
4-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
2-methyl-1-[1-(thiophene-3-carbonyl)azetidin-3-yl]piperidine
2-[1-(cyclohexylmethyl)-4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
1-cyclohexyl-4-(pyrazine-2-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]oxane-2-carboxamide
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
4,6-dimethoxy-2-[(E)-2-phenylethenyl]pyrimidine
N-[2-(2,4-difluorophenyl)-1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methylpropanamide
N-(3,4-difluorophenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
4-(1H-imidazol-1-yl)-1-(quinolin-4-yl)piperidine-4-carboxylic acid
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
3-[2-(dimethylamino)ethyl]-3-ethyl-1-(quinolin-6-yl)urea
2-[2-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]piperidine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-ethyl-N-(2-methoxyethyl)acetamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
4-[6,8-dimethyl-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]-1λ6-thiomorpholine-1,1-dione
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]acetamide
3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-{1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carbonyl]piperidin-3-yl}propan-1-one
5-{[(2-methylphenyl)methyl](2-methylpropyl)carbamoyl}thiophene-2-carboxylic acid
1-ethyl-3-methyl-4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-1H-pyrazole
2-methyl-7-{5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2,7-diazaspiro[4.4]nonane
3-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[benzyl(methyl)amino]-3-[4-({[(2-fluorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-hydroxyethyl)-N-[4-(2-methylphenyl)phenyl]-3-oxopiperazine-1-carboxamide
4-[(2,4-dimethylphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}piperidin-2-one
[2H-1,3-benzodioxol-5-yl(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methyl]dimethylamine
N-[(2,3-difluorophenyl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-hexyl-8-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-(propan-2-yloxy)benzamide
N-cyclopentyl-4-(4-{[2-(3-methoxyphenyl)ethyl]amino}piperidin-1-yl)benzamide
2,4-dimethyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrimidine-5-carboxamide
2-(furan-2-yl)-5-[1-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1H-1,2,3-triazol-4-yl]pyrimidine
1-{7,7-dimethyl-5-[(thian-4-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
4-[(2S)-2-hydroxy-2-phenylacetyl]-1-phenylpiperazin-2-one
6-[3-(1H-indol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
methyl 2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-6-[1-(methylsulfanyl)propan-2-yl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2,3-difluorophenyl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(3S,4R)-1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
(3R,4S)-4-cyclopropyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrrolidin-3-amine