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ethyl 1-{[1-(7-chloroquinolin-4-yl)-4-(ethoxycarbonyl)-1H-pyrazol-5-yl]methyl}piperidine-4-carboxylate
N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-[2-(ethylsulfanyl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
3,6-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-benzofuran-2-carboxamide
1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(propan-2-yl)-1,4-diazepane
2-(2-chlorophenyl)-N-(2-methanesulfonylethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]pyrrolidin-3-ol
N-[1-(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(oxan-4-yl)acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]propan-1-one
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[(2-chlorophenyl)methyl]-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
5-methyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-phenyl-N-[1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
1-(2-chloro-4-fluoro-5-methylphenyl)-3-methyl-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
5-acetyl-2,4-dimethyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrrole-3-carboxamide
4-{4-[(4-fluorophenyl)methyl]piperazin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(2R,3R)-1'-(2H-1,3-benzodioxol-5-ylmethyl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]acetamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
3-(3-methoxyphenyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
1-[(1-benzylpyrrolidin-3-yl)methyl]-1-methyl-3-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(pyridin-3-yloxy)acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,2-oxazol-5-ylmethyl)acetamide
2-(4-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
(3R,4R)-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
{1-[3-({[(2-fluorophenyl)methyl]amino}methyl)-7-methoxyquinolin-2-yl]piperidin-3-yl}methanol
2-(2-methoxyethyl)-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
6-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(3aS,6aS)-2-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-phenyl-N-{[1-(pyrazin-2-yl)piperidin-3-yl]methyl}benzamide
methyl 8-[(6-methylpyridin-2-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(4-chlorobenzoyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
1-[2-(4-chlorophenyl)ethyl]-N-[(2,6-difluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2,4-trimethylbenzamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-(4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
2-cyclopentyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}acetamide
3,5-dimethyl-1-({3-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]phenyl}methyl)-1H-pyrazole
5-(2-methoxyphenoxymethyl)-N-methyl-N-(3-methylbutyl)-1H-pyrazole-3-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(methoxymethyl)cyclopropyl]-N-methylbenzamide
(1S,5R)-3-benzoyl-6-(2-chlorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(9H-purin-6-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrimidin-2-amine
(2S,4R)-N-methyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N,N-dimethyl-2-({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl}amino)ethane-1-sulfonamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide