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N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3-(trifluoromethyl)benzamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)propanamide
1-[4-(3-fluorophenyl)benzoyl]-4-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
4-chloro-2-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
2-methyl-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}pyrimidine
1-{3-[1-(2-hydroxyethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]phenyl}ethan-1-one
3-(2-methoxyethyl)-5-(2-propyl-1,3-thiazol-4-yl)-1,2,4-oxadiazole
1-[({[4-fluoro-3-(trifluoromethyl)phenyl]methyl}carbamoyl)methyl]piperidine-4-carboxamide
methyl 3-({1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidin-3-yl}formamido)propanoate
2-(2-methoxyphenyl)-5-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}pyrimidine
9-(1H-1,3-benzodiazole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,5S)-1-cyclohexyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
N-[(3-fluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[7-(2,6-difluorobenzenesulfonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1,5-dimethyl-2-phenyl-4-(1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazol-2-yl)-2,3-dihydro-1H-pyrazol-3-one
3,5-dimethyl-N-(3-methyl-1-{7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(pyridin-2-yl)acetyl]-1,4-diazepan-5-one
1-{1'-[(2-butyl-1H-imidazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(2-methylphenyl)propan-1-one
(4aS,7aR)-1-[5-(3-methoxyphenyl)furan-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[4-(1H-indol-2-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
1-ethyl-8-(2-phenylethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
N'-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]butanediamide
(2S,6S)-4-methyl-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-cyclopropyl-N-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-2-phenylethyl}pyridine-2-carboxamide
3-{ethyl[(5-methoxy-1H-indazol-3-yl)methyl]amino}-1λ6-thiolane-1,1-dione
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,4-diazepane
1-ethyl-5-oxo-N-[2-(1,3-thiazol-4-yl)ethyl]pyrrolidine-3-carboxamide
2-(3-methoxypropyl)-9-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
1-[(3-methoxyphenyl)methyl]-3-methyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
2-[(3-chlorophenyl)methyl]-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-(4-fluorophenyl)-2,2-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}cyclopropane-1-carboxamide
(5S,9aS,9bS)-5-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-8-chloro-2-(furan-2-yl)quinoline
2-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1-benzofuran-5-carboxamide
6-(2-methoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]pyridazin-3-amine
{[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}dimethylamine
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-2-(4-methylpiperazin-1-yl)pyrimidine
N-[1-(2-{4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
3-methyl-8-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-(propan-2-yl)propanamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-[4-(trifluoromethyl)phenyl]urea