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5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-[3-(propan-2-yloxy)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopentyl-3-(3-hydroxy-3-methylbutyl)benzamide
4-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-[3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
4-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-hydroxybutanamide
N-(1-ethyl-1H-pyrazol-4-yl)-4-(2-phenoxyacetyl)piperazine-1-carboxamide
3-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-2-yl}pyridine
5-(2-methoxyphenoxymethyl)-N-(3-methylbutan-2-yl)-1H-pyrazole-3-carboxamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N-cyclopropyl-3-[5-(5-ethylthiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
3-methoxy-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
5-ethyl-4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-1,3-oxazole
6-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-N-(2-methoxyethyl)-8-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(piperidine-1-carbonyl)piperidine
1-[1'-(2-chlorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
(4aS,7aR)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-8-[2-(phenylamino)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}pyridin-2-ol
4-{5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(pyrrolidin-1-yl)butan-1-one
5-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-(2-methoxyethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazole
(4aR,7aS)-1-acetyl-4-[2-(propan-2-yl)pyrimidine-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2,6-dimethylphenol
N-({3,5-dimethoxy-4-[2-(1-methylpyrrolidin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-2-carboxamide
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-4-(thiophen-2-yl)butanamide
2-(1H-imidazol-4-ylmethyl)-6,7-dimethoxy-1-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
2,2,6,6-tetramethyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}piperidine
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]acetamide
N-(1-cycloheptylpiperidin-3-yl)-2-methylpropanamide
2-(2-{6-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}ethyl)-3,4-dihydroquinazolin-4-one
2-({2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}amino)-6-methyl-3,4-dihydropyrimidin-4-one
N-(2,5-difluorophenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
methyl 3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2-methyl-1,3-thiazol-4-yl)-N-[(4-phenylmorpholin-2-yl)methyl]acetamide
N-[(1-hydroxycyclohexyl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
(3S,4R)-N,N-dimethyl-1-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-4-(propan-2-yl)pyrrolidin-3-amine
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-[1-(thiophen-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
4-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
7-fluoro-3-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-benzofuran-2-carboxamide
2-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
2-{[5-({ethyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)pyrimidin-2-yl]amino}acetic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-{5-[3-(1H-pyrrol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one