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N-(4-methoxyphenyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-amine
4-(2H-1,3-benzodioxol-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-{1-[1-(2-hydroxy-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-cycloheptyl-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
{[1-(1H-1,3-benzodiazol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amine
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
(1s,4s)-N-{3-[ethyl(methyl)amino]-2-methylpropyl}-4-hydroxycyclohexane-1-carboxamide
2-phenyl-5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
1-{4-[(3-ethoxy-2-hydroxypropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
N-[(5-ethylpyridin-2-yl)methyl]-8-fluoro-N-methylquinoline-2-carboxamide
5-amino-3-(3,5-dimethyl-1H-pyrazol-4-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-ethyl-5-[2-(4-fluorophenyl)piperidine-1-carbonyl]pyrimidin-2-amine
8-(1-aminocyclopropanecarbonyl)-3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-ethyl-2-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-3-yloxy)acetamide
5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyridine-3-sulfonyl)piperidin-3-yl]propanoic acid
1-methyl-5-(3-phenylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-1,2-oxazole-3-carboxamide
ethyl 4-[4-(4-{[2-(pyridin-3-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
5-methyl-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-methyl-6-({4-[4-(1,2-oxazolidine-2-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
5-{3-[4-(2-hydroxyphenyl)piperazin-1-yl]-3-oxopropyl}-5-[(4-phenylphenyl)methyl]pyrrolidin-2-one
1-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
6-[1-(4-chlorophenyl)cyclopropanecarbonyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl 1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-4-carboxylate
methyl 5-({2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]acetamido}methyl)furan-2-carboxylate
5-(1-acetylpyrrolidin-2-yl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
N,N-diethyl-1-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxamide
3-{2-oxo-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}-4-(2-phenylethyl)piperazin-2-one
4-({4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)benzonitrile
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2-oxopyrrolidin-1-yl)propanamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-ethyl-3-(morpholine-4-carbonyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-methyl-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}pentane-1,2-dione
methyl 1-benzyl-3-cyclopropaneamido-5-[(1-methoxypropan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 1-benzyl-5-[(3-methylbutyl)amino]-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{1-methyl-4-[(5-methylfuran-2-yl)methyl]-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
5-[2-(1H-imidazol-4-yl)ethyl]-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3,5-dimethoxybenzamide
2-[2-(4-chlorophenyl)morpholin-4-yl]-N-(propan-2-yl)pyridine-4-carboxamide
6-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[(2-fluorophenyl)methyl]-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
2-(4-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
N-[(4-methoxyphenyl)methyl]-2-(1-methylpyrrolidin-2-yl)-N-(pyridin-2-ylmethyl)acetamide
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-(1-propylpiperidin-4-yl)propanamide
3-[1-(2-aminoacetyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 4-{2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(propan-2-yloxy)ethan-1-one