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N-{2-[2-(2-methoxypyrimidin-5-yl)-1H-imidazol-1-yl]ethyl}-3-methylpyridin-4-amine
N-{[1-(dimethylamino)cyclohexyl]methyl}-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[(4-methoxyphenyl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(oxolan-2-ylmethyl)acetamide
2-{[1-(2-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}cyclopentan-1-one
5-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
methyl 6-[(2,4-dimethylphenyl)methyl]-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(R)-[1-(2-methylpyridin-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl](phenyl)methanol
(3S)-1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}pyrrolidin-3-amine
2-(azepan-1-yl)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
N-({7-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-(4-fluorophenyl)ethyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
1-(oxane-2-carbonyl)-4-(pyridin-4-yl)piperazine
2-(4-fluorophenyl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
5-[1-(3-methylbenzoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
5-chloro-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-3-methyl-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
2-phenyl-4-(thiophene-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{4-[(6-chloroquinolin-2-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
(3R,4R)-3,4-dimethyl-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
4-(4-methanesulfonylphenyl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
N4-[3-(2,4-dimethylphenoxy)-2-hydroxypropyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-[2-(furan-2-yl)ethyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
5,6-dimethyl-2-{2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
1-(3,4-difluorophenyl)-3-[1-(methoxymethyl)cyclopentyl]urea
N-ethyl-2,3,6-trimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]quinoline-4-carboxamide
methyl({[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl})[1-(pyridin-3-yl)propyl]amine
(2R,3S,6R)-5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
2-methyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide
3-[(3R,4S)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
methyl 1-({4-[3-(3,5-dimethylphenyl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
N-cyclopropyl-5-[(diethylcarbamoyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-fluoro-1-methyl-2-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1H-indole
(3S,4R)-1-(1-methyl-1H-indole-4-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-{2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}morpholine
(4aS,7aR)-1-pentyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{4-phenyl-1-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl}phenol
3-[2-(2-fluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidine
3-{methyl[2-(methylcarbamoyl)ethyl]sulfamoyl}-N-(2,2,2-trifluoroethyl)benzamide
6-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-N-(propan-2-yl)pyrimidin-4-amine
N-[4-(2-fluorophenoxy)phenyl]-1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidine-4-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
(3S,4S)-1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
2-(2-butoxy-3-methoxyphenyl)-1H-1,3-benzodiazole-5-carbonitrile
2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
2-(furan-2-yl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-oxoacetamide