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1-methyl-5-[methyl(thiophen-2-ylmethyl)amino]-N-[2-(piperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(3-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2S)-1-cyclohexyl-3-hydroxypropan-2-yl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(2-oxopyrrolidin-1-yl)propanamide
(3R,4S)-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(3-methoxyphenyl)pyrrolidin-3-amine
4-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]-1-phenylpiperazin-2-one
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
N,N-dimethyl-6-{4-[(5-propylfuran-2-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
7-(3-methylfuran-2-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-ethyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1H-pyrazole-3-carboxamide
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl](1-phenoxypropan-2-yl)amine
1-[2-oxo-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethyl]azepan-2-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
(4aS,8aR)-6-(2-chlorobenzoyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-methyl-5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
1-(7-methoxy-4-methylquinazolin-2-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}piperidine-4-carboxamide
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]naphthalene-1-carboxamide
N-(2-{5-[(2,3-dihydroxypropyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(2-methoxyphenyl)propanamide
2-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-[2-(adamantan-1-yl)ethyl]-N,1-dimethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-[4-(2-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}azepan-2-one
N-[2-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-N'-(4-methylphenyl)propanediamide
2-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}pyrrolidine-1-carboxamide
methyl 1-(3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-2-carboxylate
(1S,5R)-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridin-3-yl}ethan-1-one
6-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-(3-hydroxypropyl)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-2-oxo-N-(prop-2-en-1-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
4-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)benzamide
ethyl 3-[(3-chlorophenyl)methyl]-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidine-3-carboxylate
3-[2-(azocan-1-yl)-2-oxoethyl]-1-(2H-1,3-benzodioxol-5-ylmethyl)-3-phenylpyrrolidine-2,5-dione
methyl 3-(4-cyclohexyl-1,4-diazepane-1-carbonyl)benzoate
1-{4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-4-[(2-hydroxyethyl)sulfanyl]benzamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)propanamide
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-(oxolan-2-ylmethyl)-1-(3-phenylpropyl)-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 4-(2-{[(3-chlorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carboxylate
5-propyl-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-yl]-N-(propan-2-yl)propanamide
3-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-(pyridin-2-yl)pyrimidine
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-[3-(morpholin-4-yl)propanoyl]piperidine-3-carboxylate
(1S,5R)-3-(2-amino-6-methylpyrimidin-4-yl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one