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N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopentanamine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-fluoro-N-{2-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}benzamide
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
(1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)(2-methoxyethyl)(pyridin-3-ylmethyl)amine
N-{1-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methylcyclobutanecarboxamide
3-[2-({[3-(4-chloro-1H-pyrazol-1-yl)propyl]carbamoyl}amino)phenyl]-N-methylpropanamide
2-[(4-acetylpiperazin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-({4-[(2,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
1-[2-(pyrrolidin-1-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-(2H-1,3-benzodioxol-5-yl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-methyl-3-(5-methylthiophen-2-yl)-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1H-pyrazole-5-carboxamide
3-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-1,3-oxazolidin-2-one
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
(4S)-4-acetamido-5-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-5-oxopentanamide
1-(methoxymethyl)-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}cyclobutane-1-carboxamide
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-methylfuran-3-carboxamide
3-fluoro-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
8-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-cyclopropyl-4-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrrolidin-2-one
3-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-(1-methyl-1H-pyrazol-5-yl)urea
3-(2-ethylbutyl)-8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(2,2-dimethyloxan-4-yl)methyl](methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-[2-(1H-imidazol-1-yl)ethyl]pyrrolidine-2-carboxamide
4-amino-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
3-[1-(5-amino-1H-pyrazole-3-carbonyl)piperidin-4-yl]-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-4-(4-fluorophenyl)-1-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidine-3-carboxylic acid
N-[(3-fluorophenyl)methyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-[(2-methoxy-3,5-dimethylphenyl)methyl]azetidine-3-carboxylic acid
methyl 3-(4-fluorobenzenesulfonamido)-5-[(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylformamido)methyl]benzoate
1-cyclopentyl-4-{[5-(2-ethoxyacetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperazin-2-one
2-chloro-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}pyridine-4-carboxamide
(1R,5S,6S)-6-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
(3aS,6aS)-1-oxo-2-propyl-5-[3-(pyridin-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[5-(piperidine-1-carbonyl)pyridin-2-yl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-(2,5-dimethoxyphenyl)-3-[1-(thian-4-yl)piperidin-4-yl]urea
3-(1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
4-(4-chlorophenyl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]butanamide
2-(3,4-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[1-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
2-{1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}-1,3-benzoxazole
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
5-benzenesulfonamido-N-benzyl-1-ethyl-N-(2-hydroxyethyl)-2-methyl-1H-1,3-benzodiazole-7-carboxamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide