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N-(3-cyclopentylpropyl)-N-methyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
5-(2H-1,3-benzodioxol-5-yl)-3-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
8-methyl-6,9-dioxo-N-(trimethyl-1H-pyrazol-4-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-(prop-2-yn-1-yl)-N-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}cyclohexanamine
3-(but-2-yn-1-yl)-5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}cyclohexanecarboxamide
1-(5-chloropyridin-2-yl)-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazine
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
1-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
4-(2-methoxyacetyl)-N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1,4-diazepane-1-carboxamide
9-methoxy-3-[(4-methoxy-2,3-dimethylphenyl)methyl]-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
4-methyl-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}-1,2,3,6-tetrahydropyridine-1-carboxamide
4-(2,5-dimethoxyphenyl)-2-{[(3-ethoxypropyl)amino]methyl}phenol
[2-(2-methoxy-6-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}phenoxy)ethyl]dimethylamine
N-[(3S,4R)-1-(furan-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-cyclohexyl-5-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}pyrimidine
1-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-(azocan-1-yl)propan-2-ol
2-(3-methoxypropyl)-9-[2-(methylamino)pyridine-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
[5-({3-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)furan-2-yl]methanol
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)quinoxaline-6-carboxamide
1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(pyrimidin-2-yl)-1,4-diazepane
(1R,5S)-6-({2-[(2-methylphenyl)methoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonane
8-(4-chloro-2-hydroxybenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methanesulfonyl-4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-diazepane
(1S,3R)-3-amino-N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]cyclopentane-1-carboxamide
1-[(3-methoxyphenyl)methyl]-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
6-[1-(2-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{2-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{2-[3-cyclopropyl-1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
N-ethyl-N-(2-methoxyethyl)-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-amine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-ethyl-1-({1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)urea
3-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine
6-{3-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
3-fluoro-4-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)-1-propylpyrrolidin-2-one
N-[3-(4-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-methylthiophene-2-carboxamide
3-{[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
N1-(5-methylpyridin-2-yl)-N3-(4-methylpyrimidin-2-yl)propane-1,3-diamine
3-methyl-6-[5-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,4-oxadiazol-3-yl]pyridazine
methyl 5-{[1-(4-fluorophenyl)propan-2-yl]amino}-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2-hydroxyphenyl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-(5-methylpyrimidin-2-yl)-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
[(2-ethylpyrimidin-4-yl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
(6-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridin-2-yl)methanol
2-methyl-4-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrimidine-5-carboxamide