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8-(butan-2-yl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(diethylamino)-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-cyclopentyl-5-[4-(methoxymethyl)piperidine-1-carbonyl]piperidin-2-one
N,N-diethyl-1-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(4-{[(3,4-dimethoxyphenyl)methyl](methyl)amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
2-phenyl-N-[4-(pyridin-2-yl)butyl]imidazo[1,2-a]pyridine-6-carboxamide
1-{3-[4-(benzyloxy)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
N-{2-[1-(3,3,3-trifluoropropyl)piperidin-3-yl]ethyl}pyrimidine-4-carboxamide
3-methoxy-4-{1-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-imidazol-2-yl}phenol
N,N-dimethyl-3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
N-[(3R,4S)-4-cyclopropyl-1-(3-hydroxypropyl)pyrrolidin-3-yl]-3-(2-oxoazepan-1-yl)propanamide
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]quinoline
N-cycloheptyl-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-methyl-N-{2-[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
2-{2-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-1H-imidazol-1-yl}-5-methylphenol
1-[4-(2,4-difluoro-3-methoxybenzoyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(9H-purin-6-yl)piperidin-4-amine
7-cyclopropanecarbonyl-N-[3-(1H-imidazol-1-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2-methoxyethyl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)piperidine-3-carboxamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(trifluoromethyl)benzamide
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-3-yl}propanamide
N-cyclopropyl-3-{1-[3-(morpholin-4-yl)benzoyl]piperidin-4-yl}propanamide
2-(1H-1,2,3-benzotriazole-5-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
4-({2-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
methyl 9-(cyclopentyloxy)-3-[4-(4-fluorophenyl)-4-oxobutanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
methyl 2-{[2-(phenoxymethyl)-1,3-oxazol-4-yl]formamido}acetate
N,1,3-trimethyl-N-{1-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-5-carboxamide
4-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-yl}thiomorpholine
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(ethyl)(oxolan-2-ylmethyl)amine
1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(3S)-1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)pyrrolidin-3-yl]acetamide
N-{4-[4-(but-2-ynamidomethyl)-5-methyl-1,3-oxazol-2-yl]phenyl}-5-(methoxymethyl)thiophene-2-carboxamide
N-[4-(propan-2-yl)phenyl]-1-(quinoxaline-5-carbonyl)piperidin-3-amine
5-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
9-methoxy-3-[(4-methoxy-2,5-dimethylphenyl)methyl]-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-cyclopropyl-2,3-dimethyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)-1H-indole-7-carboxamide
4-(4-fluorophenoxy)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine-4-carboxylic acid
methyl 3-(furan-2-amido)-1-methyl-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[2-(1H-imidazol-4-yl)ethyl]piperidin-4-amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-methoxy-1H-indole-2-carboxamide
N-{2-[5-methyl-4-({methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-1,3-oxazol-2-yl]phenyl}thiophene-3-carboxamide
4-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
2,3-dimethyl-N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}-1H-indole-7-carboxamide
4-{3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]phenyl}-2-methylbutan-2-ol