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N-cyclopentyl-N'-[2-(3-hydroxy-4-methoxyphenyl)ethyl]butanediamide
ethyl 2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-2-yl)acetate
5,6-dimethoxy-2-[(4-methoxypyridin-2-yl)methyl]-1,2-dihydroisoquinolin-1-one
1-(cyclopropylmethyl)-5-(2-phenoxypropanoyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2-methylphenyl)methyl]-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
(3aS,7aR)-2-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-(2,5-dioxoimidazolidin-4-yl)-N-(2-hydroxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
9-(4-methylbenzoyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
3-chloro-6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyridine-2-carboxylic acid
2-butyl-5-[4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3-benzoxazole
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-sulfonamide
{4-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1,4-oxazepan-6-yl}methanol
4-(pyridin-2-ylmethyl)-11-({[2-(trifluoromethyl)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-ethyl-5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]pyrimidine
4-(2-methyl-1H-imidazol-1-yl)-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
(1R,7S)-3-[(3-methylphenyl)methyl]-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one
N-({8-[(2-chlorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
methyl[(2-phenyl-1,3-oxazol-4-yl)methyl][1-(pyridin-3-yl)ethyl]amine
4-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]benzonitrile
N-[(1-benzylpiperidin-3-yl)methyl]cyclopentanamine
6-chloro-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1-methyl-1H-indol-3-yl)methyl]piperazin-2-yl}ethan-1-ol
4-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)-2-(4H-1,2,4-triazol-4-yl)pyridine
1-[(4-chlorophenyl)methyl]-N-[3-(morpholin-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(3-methoxypropyl)piperidine
N-ethyl-2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)furan-3-carboxamide
N-[(3,5-dimethyl-1H-indol-2-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
9-(2-oxoimidazolidine-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 3-[(3-chlorophenyl)methyl]-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-3-carboxylate
(1S,4S)-5-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-{[3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
6-fluoro-4-(4-hydroxy-4-phenylpiperidine-1-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
methyl[(5-methylfuran-2-yl)methyl]{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
9-methoxy-N-(3-methylbutyl)-7-oxo-3-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 4-[7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
ethyl 3-[(2-fluorophenyl)methyl]-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate
3-({2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-(2,6-difluorophenoxymethyl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
1-methyl-2-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}azepane
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(3aR,6aR)-2-benzyl-N-methyl-N-(pyrazin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[4-(2-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-oxoethoxy)phenyl]propanamide