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3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(3S)-2-oxoazepan-3-yl]propanamide
N-{[2-(azepan-1-yl)-7-chloroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]furan-2-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[4-(dimethylamino)phenyl]ethan-1-one
4-{3-[2-(azetidin-1-ylmethyl)phenoxy]propyl}morpholine
[(2S,4R)-4-{[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}-1-methylpyrrolidin-2-yl]methanol
3-(dimethylamino)-N-(4-methoxy-3-propanamidophenyl)pyrrolidine-1-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-5-methyl-6-(thiomorpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
3-methoxy-1-{2-[4-(2-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
2,5-difluoro-N-(1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-{1-[2-(benzyloxy)ethyl]piperidin-4-yl}methanesulfonamide
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-[3-(dimethylamino)-2,2-dimethylpropyl]propanamide
3-[(oxan-4-yl)sulfamoyl]-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
3-(3-methylbut-2-en-1-yl)-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
5-[4-(2,6-dimethylphenyl)phenyl]-1H-1,2,3,4-tetrazole
N-{[7-(2-methylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}cyclopropanecarboxamide
5-methanesulfonyl-2-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrimidin-4-amine
1-(cyclohexylmethyl)-4-[(5-ethyl-2-methylpyrimidin-4-yl)amino]pyrrolidin-2-one
8-fluoro-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}quinoline-2-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
4-ethyl-3-{1-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-{1-[2-(2-methoxyphenyl)acetyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-methyl-2-(1-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)-1,3-thiazole
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(1H-indol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-ethyl-4-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-6-methylpyrimidine
3-(1,3-benzothiazol-2-yl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}propan-1-one
(3S,4S)-4-cyclopropyl-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
4-methyl-3-({5-[1-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]furan-2-yl}sulfanyl)-4H-1,2,4-triazole
2-(2,5-dioxoimidazolidin-1-yl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
1-{[3-(furan-2-yl)phenyl]methyl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
6-chloro-2-(2,6-dimethoxyphenyl)-1,3-benzothiazole
N-[2-(2-methoxyphenyl)ethyl]-2-{4-[4-(thiomorpholin-4-yl)piperidin-1-yl]phenyl}acetamide
7-(cyclohexylmethyl)-2-(furan-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-fluorophenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
7-(cyclopropylmethyl)-2-[4-(difluoromethoxy)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
5-fluoro-2-[5-(oxane-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
(4S)-4-hydroxy-3,3,4-trimethyl-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
4-{[6-(4-methanesulfonylphenyl)pyridin-3-yl]methyl}morpholine
(1S,5R)-3-[(2,3-dimethyl-1H-indol-7-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
3-{[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]methyl}benzamide
3-[({[3-(trifluoromethoxy)phenyl]methyl}amino)methyl]piperidin-3-ol
3-[(2,8-dimethylquinolin-4-yl)formamido]propanamide
3-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,5-dimethylpyrazine
4-methyl-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-7-(methylsulfanyl)quinolin-2-amine
2-[ethyl(oxan-4-ylmethyl)amino]-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
2-(dimethylamino)-7-[(4-methyl-1H-imidazol-2-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-benzyl-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-2-one
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
1-[2-(4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]piperazine