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(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-fluoro-2-(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
2-[1-(cyclohexylmethyl)-4-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazolidin-2-yl)propanamide
6-ethyl-N-[2-(furan-2-yl)-2-hydroxyethyl]-2-methylquinoline-4-carboxamide
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[1-(pyridin-4-yl)propyl]propanamide
9-methoxy-7-(quinolin-3-yl)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,2,3-trimethylquinoxaline-6-carboxamide
6-methyl-2-oxo-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-(2-hydroxyethyl)-1-(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
N-benzyl-N-ethyl-2-(morpholin-4-yl)-6-phenylpyridine-3-carboxamide
1-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
1-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
methyl 7-oxo-9-[3-(pyridin-4-yl)propoxy]-3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-(2-cyclohexylethyl)-2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-3-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
6-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
3-cyclopentyl-5-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
3-{[ethyl(oxan-4-ylmethyl)carbamoyl]amino}-2-methyl-N-(2-methylpropyl)benzamide
4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazole
2-({4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-6-methylpyridine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,3-dimethyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
1-[2-(1H-imidazol-4-yl)ethyl]-2-[5-(oxan-2-yl)thiophen-2-yl]-1H-imidazole
4-[(4-ethoxyphenyl)methyl]-3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]piperazin-2-one
3-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}phenol
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-ethyl-3-(piperidin-3-yl)-1-[2-(1H-pyrrol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-hydroxypyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
(3R)-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-ol
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
4-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}benzoic acid
9-(cyclohex-3-ene-1-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-[3-(2-methyl-1,3-thiazol-4-yl)-5-(4-methyl-1,3-thiazol-5-yl)-1H-1,2,4-triazol-1-yl]piperidine
5-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-4-benzylpiperazine
({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-3-methylpentane-1,2-dione
7,7-dimethyl-2-(morpholin-4-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5,6,7,8-tetrahydroquinazolin-5-amine
2-(4-chloro-2-methylphenoxy)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-({7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
2-(2-aminoethyl)-N-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}quinazolin-4-amine
2-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
8-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-8-azaspiro[4.5]decane-7,9-dione