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N-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
N-benzyl-5-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}pyrimidin-2-amine
[(3R,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(2-hydroxyethyl)-9-{[4-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,4-dimethylpyrimidine-5-carbonyl)-N-(4-fluorophenyl)piperazine-2-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(oxolan-3-ylmethyl)-1,3-oxazole-4-carboxamide
6-cyclopentanecarbonyl-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
1-(2-amino-5-methylpyrimidin-4-yl)-N-cycloheptylpiperidine-4-carboxamide
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(2-methoxyethyl)-3-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)propanamide
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(pyridin-4-yl)-1,4-diazepane
2-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}-1-methyl-1H-imidazole
(1R,5R)-6-(3,4-difluorobenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxo-N-(quinolin-4-ylmethyl)piperidine-3-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(2-phenylacetyl)piperidin-1-yl]ethan-1-one
1-(4-fluorophenyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidin-3-amine
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-1-sulfonyl)piperidine
4-[5-(2-butyl-1H-imidazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]-1-methylpiperidine
(3S,4R)-3-benzyl-4-methyl-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-ol
(2E)-1-[(4aR,8aS)-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-1-yl]-3-(2-fluorophenyl)prop-2-en-1-one
2-phenyl-1-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)ethan-1-ol
N-[(3S,4R)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
N-cyclopropyl-1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
6-methoxy-3-{[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1,2-dihydroquinolin-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
6-{methyl[2-(oxan-4-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
8-({3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)quinoline
4-hydroxy-N-[1-(pyrazin-2-yl)propan-2-yl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-(4-methoxyphenyl)propan-1-ol
N-(furan-2-ylmethyl)-3,4-dimethoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}benzamide
(1R,5R)-6-benzyl-3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,5R)-1-(2-ethylbenzoyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)piperidin-2-one
1-(2-methylpropyl)-4-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
5-[5-(1-methylazepan-2-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
3-(4-methylphenoxymethyl)-1-(oxan-4-ylmethyl)piperidine
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
N-cyclopentyl-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
2-propyl-4-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyridine
N-[(3S,4R)-1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-{5-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridin-2-yl}methanesulfonamide
(2S,4R)-4-amino-1-(3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]propan-1-one
1-(2,4,6-trimethylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one