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3-[(4aR,7aS)-4-[2-(morpholin-4-yl)-2-oxoethyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]oxane-4-carboxamide
3-(2-methoxyethyl)-5-(4-methyl-1,3-thiazol-5-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
4'-(2,2-dimethylpropyl)-1-(pentan-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}benzonitrile
N-[(3S,4R)-1-(3-cyano-6-methylpyridin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
3-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-(1-ethylpiperidin-4-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
5,7-dimethoxy-4-[2-(methylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinolin-2-one
4-[2-ethyl-7-(1,2-oxazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholine
2-{1-[(4-fluorophenyl)methyl]-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-yl}ethan-1-ol
5-[2-(aminomethyl)-1H,2H-naphtho[2,1-b]furan-7-yl]pyridine-3-carboxamide
1-[(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
1-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
{2-[2-(1-{5-[(dimethylamino)methyl]furan-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
(2-methoxy-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methanol
(1S,5R)-3-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-({1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
2-methoxy-4-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyridine-3-carbonitrile
{[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
dimethyl[2-(3-{3-[5-(morpholine-4-carbonyl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)ethyl]amine
N-methyl-6-{[(3S)-2-oxoazepan-3-yl]amino}-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
1-ethyl-1-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-(1-methyl-1H-indazol-5-yl)urea
(3aS,6aR)-5-(3,6-dimethylpyrazin-2-yl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{2-[2-(2,4-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-6-methyl-3,4-dihydropyrimidin-4-one
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
(3aR,6aR)-2-[4-(dimethylamino)benzoyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(methylsulfanyl)ethyl]-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
1-(cyclopropylmethyl)-4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}-2-methylpropanamide
1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-4-phenylpiperazine
8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(3-methoxyphenyl)-1-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}ethyl]-N-methyloxane-4-carboxamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
(4S)-1-[3-(3-fluorophenyl)benzoyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
(4aS,8aR)-6-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(4-methoxy-2,3-dimethylphenyl)-1-(3-methoxypropyl)-1H-imidazole
(3S,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(hydroxymethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)[(2,3-dimethoxyphenyl)methyl]methylamine
(E)-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-2-phenyl-N-(pyridin-4-ylmethyl)ethene-1-sulfonamide
methyl 3-(3,4-dimethylbenzoyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2-ethoxyphenyl)ethan-1-one
2-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-4-carbonitrile
3-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-1-cyclopentylurea
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
(2-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
4-(1-ethyl-3-methylpiperidine-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one