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N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-[N-(3-methylphenyl)methanesulfonamido]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
(3R,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(4-cyanonaphthalen-1-yl)-1-[(3-hydroxypiperidin-3-yl)methyl]urea
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-ethyl-N-(2,2,2-trifluoroethyl)acetamide
(2E)-1-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
(3S)-3-ethyl-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)morpholine
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
5-(2H-1,3-benzodioxol-5-yl)-3-cyclopentyl-1-ethyl-1H-1,2,4-triazole
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})amine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrrolidine-3-carboxamide
3-(2-fluorophenyl)-1-methyl-3-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
2-[benzyl(methyl)amino]-N-(2-hydroxyethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-[1-(4-methanesulfonylphenyl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-phenoxyethan-1-one
(4-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-oxazepan-6-yl)methanol
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-5,6-dimethylthieno[2,3-d]pyrimidin-2-yl}ethan-1-amine
2-{1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
4-{6-[2-(pyridin-3-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
6-[(diethylamino)methyl]-N-(piperidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2R,3R)-1'-benzyl-3-(1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-3,5-dimethyl-1H-pyrrole-2-carboxamide
1-{[4-(2-aminoethyl)phenyl]methyl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
methyl 4-(5-{[(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
5-chloro-N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-3-fluoropyridin-2-amine
5-({[(3-{2-[4-(2-fluorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
4-[5-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)furan-2-yl]benzoic acid
1-ethyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1H-pyrazole-4-sulfonamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-N,N-dimethylpiperazine-1-carboxamide
N-methyl-5-(naphthalen-1-yl)-N-[2-(oxan-4-yl)ethyl]-1,2,4-triazin-3-amine
1-[2-({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)ethyl]piperidin-2-one
3-phenyl-8-{thieno[2,3-d]pyrimidin-4-yl}-1,8-diazaspiro[4.5]decan-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
1-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
7-[(2,3-difluorophenyl)methyl]-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
(1R,7S)-N-benzyl-N-methyl-4-oxo-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-{1-[5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-yl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-ethyl-3-{2-[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
4-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}thiomorpholine
4-[3-(7-cyclobutanecarbonyl-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
N-methyl-5-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 4-{5-chloro-2-[(cyclobutylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
3-[(3R,4S)-1-[(1-methyl-1H-indol-6-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid