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[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl}){[3-(methylsulfanyl)phenyl]methyl}amine
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-N-methylpyridine-3-carboxamide
methyl 5-{[(4-ethoxyphenyl)methyl]amino}-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
5-(2-methoxy-4-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(benzyloxy)-8-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
(5S,9aS,9bS)-5-(3,5-difluorophenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)pyridine-2-carboxylic acid
2-[5-(1-phenylcyclopropanecarbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-(5,6-dimethylpyrazin-2-yl)pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-(2-fluorophenyl)-3-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
1-(3-methylbutyl)-N-(2-methylpropyl)-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
8-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-benzyl-4-hydroxypiperidin-1-yl)-3-(1-methylpiperidin-2-yl)propan-1-one
2-{1-[(4-ethoxyphenyl)methyl]-4-(quinolin-4-yl)piperazin-2-yl}ethan-1-ol
5-cyclobutanecarbonyl-1'-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(4-fluorophenyl)-4-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]butanamide
(4aR,8aR)-7-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
3-chloro-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}thiophene-2-carboxamide
4-(4-fluorophenoxy)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
2-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-6-methylquinolin-4-ol
N-{1-[4-(4-hydroxypiperidine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}-2,4-dimethylbenzamide
9-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-{1-[3-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}piperidin-4-ol
4-(benzyloxy)-1-(1H-pyrrole-2-carbonyl)piperidine
3-(3-methylpiperidin-1-yl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
3-[5-(3-phenyl-1,2,4-oxadiazol-5-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[1-(4-methanesulfonylphenyl)propyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-11-({[4-(trifluoromethoxy)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
9-[(2S)-2,4-diaminobutanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-phenoxypiperidine-4-carboxylic acid
N-methyl-1-[(2-methylphenyl)methyl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
4-hydroxy-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N,N,2-trimethyl-3-({[3-(pyridin-4-yl)propyl]carbamoyl}amino)benzamide
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-3,3-dimethylcyclohexan-1-amine
3-(morpholine-4-sulfonyl)-5-(pyrimidin-5-yl)benzoic acid
(1S,5R)-6-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-[(4-fluorophenyl)methyl]-N-methyl-1,2-oxazole-5-carboxamide
5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide
5-[(1S,3R)-3-aminocyclopentaneamido]-N,N-dimethyl-1-benzothiophene-2-carboxamide
[5-({3-[2-(1-benzofuran-2-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)furan-2-yl]methanol
1-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}cyclopropane-1-carboxamide
(2S)-3-(4-hydroxyphenyl)-2-({1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazol-4-yl}formamido)propanamide
2-[4-({4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenoxy]ethan-1-ol