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3-(4-cyclohexylphenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrazole
N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
4-{5-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-ethyl-5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidine
(benzylsulfamoyl)({[3-(pyrrolidin-1-ylmethyl)phenyl]methyl})amine
2-methoxy-6-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}phenol
2-(2,4-difluorophenoxy)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
3-(3-methoxyphenyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
[(1-methyl-1H-pyrazol-4-yl)methyl]({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylbenzamide
2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]quinoline
3-ethyl-6-(2-phenylpyrrolidine-1-carbonyl)-3H-imidazo[4,5-b]pyridin-2-amine
N4-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5-methylpyrimidine-2,4-diamine
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
3-[({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-ethyl-5-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
3-benzyl-8-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2,4-difluorophenyl)methyl]-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
3-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1-{3-[(5-methylpyridin-2-yl)amino]propyl}urea
2-chloro-4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
2-cyclopropyl-8-[(5-propylfuran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-[2-(oxan-2-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-(3-chloro-4-methoxyphenyl)-6-(5-fluoro-1H-indole-2-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(phenylamino)pyrimidine-5-carboxamide
N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}piperidin-3-amine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-[2-chloro-5-(piperidine-1-carbonyl)phenyl]-4-methyl-1,4-diazepane-1-carboxamide
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(1H-indol-3-yl)pyridine-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2-dimethyl-1,3-benzoxazole-6-carboxamide
(3aR,6aR)-N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(1R,9aR)-1-{[methyl(quinolin-5-ylmethyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
1-(2-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}pyrimidin-4-yl)piperidin-3-ol
3-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(prop-2-en-1-yl)propanamide
methyl 3-benzamido-6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-cyclopentyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}propanamide
(3S,4S)-4-cyclopropyl-1-(1H-pyrazole-4-sulfonyl)pyrrolidine-3-carboxylic acid
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
6-[(2-hydroxyphenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-cyclopropyl-5-[2-(1H-indol-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(2-methoxyethyl)-6-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1,3-benzoxazole
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(4H-1,2,4-triazol-4-yl)benzamide
1-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]-2-phenoxyethan-1-one
4-(1-{[(4-fluorophenyl)methyl]carbamoyl}piperidin-3-yl)benzoic acid
1-(4-chloro-2-methoxy-5-methylphenyl)-3-[3-(1H-imidazol-1-yl)propyl]urea
5-chloro-3-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one