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8-(3-methyl-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-1-yl)quinoline
N-methyl-6-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,4,5,6-tetrahydropyridazine-3-carboxamide
6-{[4-(diphenylmethyl)piperazin-1-yl]methyl}-2-oxo-N-[1-(thiophen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
5-(3-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-N,N-dimethylfuran-2-carboxamide
(1S,5R)-3-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 2-(1-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}-N-methylformamido)acetate
1-methyl-2-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
(furan-2-ylmethyl)(methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-methoxy-8-[3-(5-methylfuran-2-yl)butyl]-1,8-diazaspiro[4.5]decan-2-one
1-{5-[(3-methoxyphenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-4-ol
3-[1-(4-cyanopyridin-2-yl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
4-(2-methoxyphenyl)-2-methyl-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperazine
2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
1-(2,4-dimethylphenyl)-4-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazine
3-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}propanoic acid
1-cyclopentyl-4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
4-[2-amino-3-cyano-6-(2,2-dimethylcyclopropyl)-5-methylpyridin-4-yl]benzamide
5-(2-{2-[2-(dimethylamino)ethyl]piperidin-1-yl}-2-oxoethyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(1,3-thiazol-2-yl)ethyl]-1H-indole-3-carboxamide
6-(2,2-dimethylcyclopropanecarbonyl)-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
5-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
N-[1-(hydroxymethyl)cyclopentyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
3-{1-[2-(adamantan-1-yl)acetyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
methyl 4-{[2-(benzyloxy)phenyl]carbamoyl}piperazine-1-carboxylate
2-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
5-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-[2-(4-chlorophenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
2-(4-fluorophenoxymethyl)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
5-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydroisoquinoline
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2-methoxyphenyl)-3-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]propanamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methoxyhexan-1-one
N-(1-methoxybutan-2-yl)-4-(4-methylphenoxy)piperidine-4-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1,3,6-tetramethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-methoxy-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}quinoline
5,8-difluoro-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,2,3,4-tetrahydroisoquinoline
4-{[(1-ethyl-1H-imidazol-2-yl)methyl]amino}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N,N-dimethylacetamide
5-methyl-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-amine
(4aS,8aR)-6-{furo[3,2-c]pyridin-4-yl}-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
N-[(2S,4R,6S)-2-ethyl-6-{3-methylimidazo[1,5-a]pyridin-1-yl}oxan-4-yl]benzamide
1-cyclohexyl-4-(2,4-dimethoxybenzoyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[2-(thiophen-2-yl)acetyl]piperidin-3-yl}propanamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(4-oxo-4-phenylbutanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide