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7-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-methyl-N-[(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
4-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]piperazine-1-carboxamide
2-(3,5-difluorophenyl)-N,N-dimethylpyridine-3-carboxamide
2-(1-methyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-(3-methoxyphenyl)-1-(thiophene-2-carbonyl)piperidine
1-propyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]piperidin-4-amine
1,6-dimethyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
5-(4-methyl-1,4-diazepan-1-yl)-2-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-2,3-dihydropyridazin-3-one
2-ethyl-8-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N,8-dimethyl-3-{[methyl(oxan-4-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-{6-hydroxy-4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1,4-diazepan-1-yl}-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
4-ethyl-1-methyl-3-{1-[4-(morpholin-4-yl)butanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
2-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
5-{4-phenyl-1-[2-(thiophen-2-yl)ethyl]-1H-imidazol-5-yl}pyrimidin-2-amine
3-[(3R,4S)-1-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
5-[(2-chlorophenyl)methyl]-5-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
3-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}adamantan-1-yl acetate
4-(3-ethyl-1,2-oxazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(4-carbamoyl-3-chlorophenyl)-5-chloropyridine-3-carboxylic acid
1-{3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
1-(2,8-dimethylquinoline-4-carbonyl)-N,N-dimethylazepan-4-amine
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
ethyl 2-{[5-({[(4-methanesulfonylmorpholin-2-yl)methyl]amino}methyl)pyrimidin-2-yl](methyl)amino}acetate
3-(1H-1,3-benzodiazol-2-yl)-N-(1-cyclobutanecarbonylazepan-3-yl)propanamide
1-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
N,2,7-trimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-cyclopropyl-1,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-2,3-dihydro-1H-indene-2-carboxamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
2-(1H-indol-1-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[2-(dimethylamino)ethyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
5-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-(5-chloro-2-fluoro-4-methylphenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
5-(2,6-dimethoxyphenyl)-1-(2-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
1-benzyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrrolidin-3-amine
(1R,5R)-10-[4-(3-hydroxy-3-methylbutyl)benzoyl]-3,7,10-triazatricyclo[3.3.3.01,5]undecane-2,6-dione
{1-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-4-ylmethyl)amine
1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(2-methoxy-5-phenylphenyl)urea
methyl 3-[(4-methoxy-2,3-dimethylphenyl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(3,4-dimethoxyphenyl)-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)propanamide
4-({4-[3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
5-[5-(2-chlorophenyl)furan-2-carbonyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[4-ethyl-6-(4-methanesulfonylphenyl)pyrimidin-2-yl]morpholine
(2S,4R)-4-amino-1-(1H-indol-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide