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N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}benzamide
3-methyl-1-{1-[6-(piperidin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
(3E)-1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-3-en-1-one
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-fluoro-1,2-dihydroquinolin-2-one
(1s,4s)-N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-4-hydroxycyclohexane-1-carboxamide
[(1,2-dimethyl-1H-imidazol-5-yl)methyl]({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
7-methyl-3-[(2,4,6-trimethoxyphenyl)methyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-(diphenylmethyl)-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-[(8-methoxyquinolin-2-yl)methyl]-1-methylpiperazin-2-one
N-[(2,3-dimethylphenyl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-phenyl-7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
[(2S)-1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
(2S)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
2-{2-oxo-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethyl}-3-phenylcyclopent-2-en-1-one
N-[1-(4-fluorophenyl)ethyl]-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
1-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-3-(pyridin-4-yl)propan-1-one
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2,4-dimethyl-N-[2-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
3-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
2-(3-methylphenyl)-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
5-[1-(4-methylphenyl)cyclopropanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-3-(pyridin-4-yl)propanamide
3,4,4-trimethyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-ol
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(quinolin-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(1R,5S,6S)-6-{4-[(4-fluorophenyl)methyl]piperazine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
5-chloro-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-4-sulfonamide
(4aS,7aR)-1-[(5-methylnaphthalen-1-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(4aR,7aS)-4-[(6-methylpyridin-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-4-oxobutane-1-sulfonamide
1-(adamantan-1-yl)-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperazine
3-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-1H-pyrazole
8-(2-hydroxy-4-methylbenzoyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(pyrimidin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
7-(6-methoxypyridin-3-yl)-3,4-dihydro-2H-1-benzopyran-4-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(1H-pyrazol-4-yl)benzamide
4-[(2,2-difluoroethyl)sulfamoyl]-N-{2-[(2R)-pyrrolidin-2-yl]ethyl}benzamide
(1-methoxypropan-2-yl)({[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl})amine
(2S,4R)-1-(adamantan-2-yl)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
4-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carbonyl}-1-(prop-2-en-1-yl)pyrrolidin-2-one
N-{3-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-{thieno[3,2-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)acetamide
(1S,9S)-11-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5-(2-chloro-4-methoxyphenoxymethyl)-3-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-1H-pyrazole
1'-(1H-indole-2-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(4-fluorophenyl)methyl]-5-{[(1-hydroxycyclohexyl)methyl]amino}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole