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3-{[ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
2-{[2-({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}(methyl)carbamoyl)phenyl]amino}acetic acid
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
1-[2-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}cyclopropanamine
N-(3,5-dimethylphenyl)-2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
2-[({2-[3-(azepan-1-yl)-2-hydroxypropoxy]-5-chlorophenyl}methyl)(methyl)amino]-N-methylacetamide
4-benzyl-3-[1-(2-methyloxolane-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(cyclopropylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
2-(4-fluorobenzoyl)-7-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
2-methyl-6-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine
3-chloro-2-[3-(1-methoxyethyl)phenyl]pyridine
4-(2,3-dihydro-1-benzofuran-2-carbonyl)-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[3-(1-phenyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
4-(4-fluoro-2-methylphenoxy)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxylic acid
2-(4-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
9-(1-benzofuran-2-ylmethyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[4-oxo-7-(2-propoxyacetyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
8-[3-amino-3-(3,4-dimethoxyphenyl)propanoyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[2-(1,3-thiazol-4-yl)acetyl]-1,4-diazepan-2-one
1-(3-methoxybenzoyl)-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazine
3-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methoxy}pyridin-2-amine
2-cyclohexyl-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}pyrimidine
(2R,3R)-3-methoxy-1'-(3-phenoxypropyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(2-chlorophenoxy)-1-(1,3-thiazol-4-ylmethyl)piperidine
N-[(2-ethoxyphenyl)methyl]-N-ethylimidazo[1,2-a]pyridine-6-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-1-methyl-1H-pyrazole-5-carboxamide
1-(2-{1-ethyl-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-1,2-dihydropyridin-2-one
3-{[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}pyridin-2-amine
1-[(4-fluorophenyl)methyl]-2-methyl-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3-(1-ethyl-1H-imidazol-2-yl)piperidine
1-({4-[(3,4-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
6-(4-chlorophenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(diphenylmethyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-{2-[2-(ethylamino)pyrimidin-5-yl]-7-fluoroquinoline-4-carbonyl}piperidine-3-carbonitrile
(2S)-2-({2-[(quinolin-8-yloxy)methyl]-1,3-oxazol-4-yl}formamido)propanamide
1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-N-[(1-methylpiperidin-4-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
(2S,4S,5R)-4-(cycloheptylcarbamoyl)-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
2-{[1-(1H-pyrazol-1-yl)propan-2-yl]amino}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-benzyl-3-(2-methylphenyl)-3-[2-(3-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
N-cyclopropyl-3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)propanamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
(4aS,7aR)-1-[3-(dimethylamino)-2,2-dimethylpropyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-propoxyethyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
[2-(2-fluoro-6-methoxyphenyl)-8-methylquinolin-3-yl]methanol