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1-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-3-yl}pyrrolidin-2-one
3-methoxy-5-{methyl[2-(1H-pyrazol-1-yl)ethyl]carbamoyl}benzoic acid
(3aS,6aS)-2-[(2-aminopyridin-3-yl)methyl]-5-(3-methoxypropanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-4-amino-1-[(dimethyl-1,3-thiazol-5-yl)sulfonyl]-N-methylpyrrolidine-2-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(6-methoxypyridin-3-yl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carboxamide
N-(pyridin-3-ylmethyl)-7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
methyl 4-oxo-4-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)butanoate
{[5-(methoxymethyl)furan-2-yl]methyl}(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-{2-[1-(4-methoxyphenyl)-1H-imidazol-4-yl]ethyl}acetamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-phenyl-N-propyl-1H-1,2,3-triazole-4-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-[(4-phenyloxan-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
{5-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
6-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
ethyl 5-({[6-oxo-1-(2-phenylethyl)piperidin-3-yl]formamido}methyl)furan-2-carboxylate
N,N-dimethyl-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butanamide
methyl 5-[(butan-2-yl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-(5-carbamoyl-2-methylphenyl)-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
4-(1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-methylpropan-2-yl)morpholine
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
6-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-ethyl-5-[(furan-2-ylmethyl)amino]-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
9-(4,6-dimethylpyridine-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
N,2-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-[3-(5-chloro-2-methoxyphenyl)-1H-indazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
ethyl 1-{[(1-benzyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-imidazole-2-carboxylate
N5-[2-(pyridin-2-yl)ethyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-{[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl}cyclopentanamine
6-({methyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)naphthalen-2-ol
1-{5-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-5-methyl-1,3,4-oxadiazol-2-amine
1-[3-(dimethylamino)-2,2-dimethylpropyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-ethyl-8-[(2E)-2-methylbut-2-en-1-yl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N3-methyl-N5-(naphthalen-1-ylmethyl)-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
[(3-methoxyphenyl)methyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
5-(1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
2-{[2-(2-hydroxyethoxy)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-methyl-4-[(5-methylfuran-2-yl)methyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(3-acetylphenyl)-3-(2,5-difluorobenzoyl)piperidine-1-carboxamide
(4aS,7aR)-1-[(3-chlorophenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(furan-2-ylmethyl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
N-{[8-(1H-indole-2-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
6-(methoxymethyl)-N,1-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine