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1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
4-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperazine-2-carboxylic acid
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,2-bis(prop-2-en-1-yl)piperidine
2-methoxy-N-{3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{4-benzyl-1-[(8-methoxyquinolin-2-yl)methyl]piperidin-4-yl}methanol
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-phenylpyrrolidine-2,5-dione
ethyl 1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
methyl 2-[6-methyl-5-(thiophene-2-sulfonamidomethyl)-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl]benzoate
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
6-{4-[(1R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]piperazine-1-carbonyl}pyridin-2-ol
(3S,4S)-1-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
methyl 4-{4-[2-(pyridin-3-yl)acetyl]piperazin-1-yl}benzoate
2-phenoxy-N-{1-[7-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
2-(oxane-4-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
(1R,2R,4R)-N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
ethyl 1-(3-methylbutyl)-5-(oxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(cyclopropylmethyl)-8-[3-(3,4-dimethylphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-methoxy-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-2-carboxamide
9-[(2-fluorophenyl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-({4-[3-(azetidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(methylsulfamoyl)ethyl]-1H-pyrazole-3-carboxamide
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)propanamide
5-methyl-4-{[1-(3-methylpyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
5-(pyridin-2-yl)-5-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(3-methoxyphenyl)-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-one
5-chloro-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
6-{[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
methyl N-{1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-oxopropan-2-yl}carbamate
2-(dimethyl-1,3-thiazol-4-yl)-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
1-(3-methoxyphenyl)-6-methyl-4-(1-methyl-1H-1,3-benzodiazole-2-carbonyl)piperazin-2-one
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
N-ethyl-5-methyl-6-(2-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
9-(4-hydroxybenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
4-[(4-methoxy-3-methylphenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-[(2R,3R)-2-ethoxy-1'-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-(2-hydroxyethyl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)benzamide
5-ethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
2-(4-acetylphenoxy)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]acetamide
(2S,4S)-1-(2,4-dimethylbenzoyl)-N,N-diethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
N-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
13-[2-(propylsulfanyl)pyrimidin-5-yl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
3-{[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
1-(2-cyclopropylquinoline-4-carbonyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one