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1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
3-methoxy-N-{[1-(pent-2-yn-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}benzamide
14-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,4-dihydroquinolin-4-one
(1s,4r)-4-butyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}cyclohexane-1-carboxamide
2-(3-{[4-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
3-(2,5-difluorobenzoyl)-1-(3-phenylpropyl)piperidine
6-[(3-methoxyphenyl)methoxy]-4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(2-phenylethyl)-1,4-diazepan-2-one
N-butyl-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
(3-cyclopentylpropyl)({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
N-(5-chloro-2-methylphenyl)-4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carboxamide
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,6-dimethylquinoline-4-carboxamide
2-ethyl-9-(morpholine-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
6-(1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
(1S,4S)-2-(2-chlorophenyl)-5-[(4-oxo-4H-chromen-3-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
3-{imidazo[1,2-a]pyridin-2-yl}-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3-(thiophene-2-carbonyl)piperidine
[(1-ethyl-1H-imidazol-2-yl)methyl]({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
4-cyclohexyl-3-{[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]methyl}-4H-1,2,4-triazole
1-(4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
2-butyl-8-[2-(propan-2-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 6-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
methyl 2-{4-[(6-chloropyridin-2-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
4-{2-[2-(dimethylamino)ethoxy]phenyl}benzonitrile
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
3-[(4aR,7aS)-4-(2,3-dimethylbenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-[(1-ethyl-1H-indol-5-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
N-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-[benzyl(methyl)amino]-3-[4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-methyl-2-[(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)methyl]-1H-1,3-benzodiazole
1-{1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[3-fluoro-5-(trifluoromethyl)phenyl]-4-(1H-pyrazol-1-ylmethyl)piperidine-1-carboxamide
5-{3-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-oxopropyl}-5-[(3,4-dimethoxyphenyl)methyl]pyrrolidin-2-one
ethyl 2-{4-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-1-yl}acetate
N-(2-chlorophenyl)-3-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)propanamide
N-(3-hydroxy-2,2-dimethylpropyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
(3aR,7aS)-2-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-[1-(thiophene-2-carbonyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-{1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperidin-4-yl}-3-phenylpropan-1-ol
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
ethyl 5-[2-(2-chloro-4-fluorophenyl)acetyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
2-(3-fluoro-4-methoxyphenyl)-4-(pyrrolidine-1-carbonyl)pyridine
N'-cyclopentyl-N-[(1R,2R,3R,5S)-2,6,6-trimethylbicyclo[3.1.1]heptan-3-yl]butanediamide