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N-[(3-methylphenyl)(phenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
6-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-2,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-(1-cycloheptylpiperidin-3-yl)-3-(4-methoxyphenyl)propanamide
5-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
N-[2-(pyrazin-2-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
(3R,4R)-4-ethyl-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine-3,4-diol
propyl (4aR,7aS)-4-(3-ethyl-1,2-oxazole-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
[(3R,4R)-1-[(2-methoxy-4-methylphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(4-fluoro-3-methoxyphenyl)methyl]-8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decane
4-(2-methyl-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-2-yl)morpholine
7-(cyclopropylmethyl)-2-[3-(4-methoxyphenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3,5,7-trimethyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
(4aS,8aR)-1-(2-aminoethyl)-6-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
5-chloro-3-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-indole-2-carboxamide
N-benzyl-N-[2-(dimethylamino)ethyl]-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
3-(3,4-difluorophenyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]propanamide
(4S,6R)-N-[2-(2-fluorophenoxy)ethyl]-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
4-(1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
2-chloro-4-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]benzamide
ethyl 1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[(2R,3R)-1'-(2,2-dimethylpropyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
7-fluoro-N,2-dimethyl-N-[3-(oxolan-2-yl)propyl]quinoline-4-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(1-phenylcyclopropyl)propanamide
N-ethyl-2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-3-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2,3-difluorobenzamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
5-cyclopropanecarbonyl-1'-(1H-indole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methoxy-2-methyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
(2S,4S)-4-amino-1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-N-methylpyrrolidine-2-carboxamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(3-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[2-(dimethylamino)ethyl]-8-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-9-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-1-[3-(morpholin-4-yl)benzoyl]-N-(2-phenylethyl)piperidin-3-amine
1-{4-[(4-chlorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-methoxypropan-1-one
2,5-dimethyl-3-{4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}pyrazine
4-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid
methyl 6-(1-hydroxypropan-2-yl)-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aS,8aR)-1-(4-hydroxybutyl)-6-[3-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-({7-[(2E)-3-(3,5-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[(3R)-4-hydroxy-3-methylbutyl]-1,2-oxazole-3-carboxamide
4-[(diethylamino)methyl]-N-(2,2-dimethyloxan-4-yl)-5-ethyl-N-methylfuran-2-carboxamide
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}pyrimidin-4-amine
N-cyclohexyl-2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-(prop-2-yn-1-yl)acetamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
N-[(2,6-difluorophenyl)methyl]-1-(6-methoxy-4-methylquinazolin-2-yl)piperidin-4-amine
1-[(1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]pyrrolidin-2-one