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5-(4-acetylphenoxymethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetamide
1-methyl-1'-[5-(propan-2-yl)pyrimidin-4-yl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[4-(2,2-diphenylacetyl)piperazin-1-yl]-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
methyl 3-(2-ethylbutyl)-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(2,4-difluorophenyl)methyl]piperidine-4-carboxylic acid
4-{1-[2-(4-methylpiperazin-1-yl)butyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
2-chloro-4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}-6-methoxyphenol
1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-[(2-chlorophenyl)methyl]-6-(3-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)piperidin-2-one
7-[(1-methyl-1H-imidazol-5-yl)methyl]-N-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}pyrrolidin-2-yl)pyridine
ethyl 1-[3-(2-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-3-carboxylate
2-(2-{[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]methyl}phenoxy)propanoic acid
3-(2-methoxyphenyl)-N-{1-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-1H-pyrazol-4-yl}propanamide
6-methyl-1-(2-methylphenyl)-4-[4-(morpholin-4-yl)benzoyl]piperazin-2-one
3-(3,4-dimethoxybenzoyl)-N-(2,6-dimethylphenyl)piperidine-1-carboxamide
2-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5,7-dimethylpyrazolo[1,5-a]pyrimidine
5-(1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-4-yl)-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
2-[4-(2-fluoro-4-methylbenzoyl)piperazin-1-yl]-4-methyl-6-(trifluoromethyl)pyrimidine
1-(3-chlorophenyl)-4-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperazin-2-one
1-[3-methoxy-4-({3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
2-{4-[(6-methylpyridin-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(2,2-dimethylpropanoyl)piperidin-3-yl]propanamide
3-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}-2,2-dimethylpropan-1-ol
2-(phenylsulfanyl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(cyclohexylmethyl)[(6-{octahydropyrrolo[1,2-a]piperazin-2-yl}-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl)methyl]amine
N-[(2R,3R)-1'-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
2-[(4-methoxyphenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
5-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
1-(3-aminoazepan-1-yl)-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
N-(1-methyl-1H-pyrazol-4-yl)-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(oxan-4-yl)piperidine
5-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-oxopropyl]-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
5-benzyl-5-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[1-(pyridin-4-yl)propan-2-yl]propanamide
{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
2-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]morpholine
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-3-carboxylate
N-(1-methyl-1H-pyrazol-5-yl)-3-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}benzamide
2-ethyl-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}pyrimidine-5-carboxamide
2-(dimethylamino)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(3-methylphenyl)acetamide
2-methyl-5-({[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-1,3,4-oxadiazole
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
ethyl({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(2-methylprop-2-en-1-yl)amine
(2R,4S)-4-hydroxy-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-2-carboxylic acid
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-amine