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2-(8-methoxy-2-methylquinolin-5-yl)pyridin-3-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-ethyl-N-(3-phenylpropyl)acetamide
2-(3-cyclopentyl-5-{2-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[2-(pyridin-3-yl)acetyl]piperidine-3-carboxylate
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
3-[5-(4-fluoro-2-methylphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-ol
1-[4-(2-methoxyethyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1H-pyrazole-4-carboxamide
2-(3-phenylpropyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-3-(2-methylphenyl)propan-1-one
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2-(3-methyl-1H-pyrazol-1-yl)acetamide
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
2-[3-(4-fluorophenoxy)propyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
4-methyl-6-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(2R,3R)-1'-(2-cyclohexylacetyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(3-methylpiperidin-1-yl)ethyl]benzamide
{2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-4-(4-fluorophenyl)-N-(2-methoxyethyl)-4-oxobutanamide
N-[2-(benzyloxy)ethyl]-1-methylazepane-2-carboxamide
{4-[(2-chlorophenyl)methyl]-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanol
(3S,4R)-1-[(1-benzyl-1H-imidazol-5-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-acetyl-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1,4-diazepane-1-carboxamide
3-[5-(propan-2-yl)pyrimidin-4-yl]benzoic acid
2-(dimethyl-1,2-oxazol-4-yl)-1-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
1-(2,5-dimethylfuran-3-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
(3S)-N,N-dimethyl-1-[2-(phenylamino)pyrimidine-5-carbonyl]azepan-3-amine
3-(4-chlorobenzoyl)-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidine
1-ethyl-N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}propan-1-one
8-[(6-chloropyridazin-3-yl)oxy]-5-(morpholin-4-ylmethyl)quinoline
2-methyl-N-[3-(5-methyl-4-{[2-(2-methyl-1H-indol-3-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-3-carboxamide
ethyl 4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperazine-1-carboxylate
(3aR,6aR)-N-[2-(benzyloxy)ethyl]-2-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(5-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
(5R)-5-[3-(2-chloro-4-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
[(1-cyclopentylpiperidin-4-yl)methyl][(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](pyridin-3-ylmethyl)amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(pyridin-3-yl)acetamide
[1-(2-methyl-1,3-thiazol-4-yl)ethyl]({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl})amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2-(2,5-dimethylphenyl)-1-(2-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)ethan-1-one
8-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1-oxa-8-azaspiro[4.5]decane
N-[2-(dimethylamino)ethyl]-4-fluoro-2-methyl-N-(thiophen-3-ylmethyl)benzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-7-one