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2-{4-[(3-cyanophenyl)methyl]morpholin-3-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
5-[1-(4-oxo-4H-chromene-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(3S,4R)-1-(2-methoxy-4-methylbenzenesulfonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
2-(2-hydroxyethyl)-9-[(4-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[2-(benzyloxy)ethyl]azetidin-3-yl}-2-methylpiperidine
N-ethyl-5-[4-(4-methoxybutyl)piperazine-1-carbonyl]pyrimidin-2-amine
1-(8-chloroquinolin-5-yl)-3-(oxolan-2-ylmethyl)urea
N-{3-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}acetamide
2-(5-fluoro-2-methoxyphenyl)-2-[4-(prop-2-en-1-yl)piperazin-1-yl]acetic acid
4-(hydroxymethyl)-N-phenyl-4-(2-phenylethyl)piperidine-1-carboxamide
5-(2,6-dimethoxyphenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
1-cyclobutanecarbonyl-4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidine
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5-(3-{4-[hydroxy(pyridin-3-yl)methyl]piperidin-1-yl}-3-oxopropyl)-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
(3S,4R)-1-(5-methylpyrazine-2-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
5-[(2-chlorophenyl)methyl]-8-ethoxy-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[2-(2-methoxyphenoxy)ethyl]-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
5-ethyl-2-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
(4aS,8aR)-1-(carboxymethyl)-6-(pyridin-4-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
(1S,5R)-6-[3-(benzyloxy)propyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-methoxyphenyl)-5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1H-pyrazole
5-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-phenyl-1H-imidazole-4-carboxamide
(2S,4R)-4-[4-({[(3-cyanophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-4-(propan-2-yl)-1,3-thiazole
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)azetidin-3-ol
2-(2,3-dimethoxy-5-methylphenyl)-N-(propan-2-yl)pyrimidin-4-amine
2-[(3-fluorophenyl)methyl]-4-{3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
6-(morpholin-4-yl)-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-4-amine
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-3-yl)acetamide
N-[(4-fluorophenyl)methyl]-3-{1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-4-yl}propanamide
3-[(3R,4S)-1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
6,7-dimethoxy-2-[1-(1H-1,2,3-triazole-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
3-(2-chlorophenyl)-1-(3-methoxypropyl)-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(morpholin-2-yl)ethan-1-one
9-(cyclopropylmethyl)-4-(5-fluoropentyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-({2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}methyl)-3-(propan-2-yl)-1,2,4-oxadiazole
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
ethyl 3-benzyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine-3-carboxylate
3-amino-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,2,4-triazole-5-carboxamide
5-[(4-methoxynaphthalen-1-yl)methyl]-5-{3-[3-(3-methylbutanoyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-3H,4H,5H,7H-thieno[3,4-d]pyrimidin-4-one
3-[methyl({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl})amino]propan-1-ol
N-cyclopropyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyridine-2-carboxamide
3-[2-(N-methylmethanesulfonamido)ethyl]-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[4-(trifluoromethoxy)phenyl]methyl}amine
2-(3-hydroxy-1,2-oxazole-5-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-{4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide