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N-({3-[(3-chlorophenyl)methyl]-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl}methyl)acetamide
N-{2-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-fluorobenzamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-2-carboxamide
2-(3-acetyl-1H-indol-1-yl)-N-[(2-ethyl-1,3-thiazol-4-yl)methyl]butanamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
3-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[5-(2-methylpropyl)thiophen-2-yl]methyl}amine
(1R,5S,6S)-6-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
5-cyclohexaneamido-N-(furan-2-ylmethyl)-1-(2-methoxyethyl)-N-methyl-1H-1,3-benzodiazole-7-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amine
N-(1-ethyl-1H-pyrazol-5-yl)-2-{4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
N-(2,5-dimethyl-3-{1-[(2R)-oxolan-2-ylmethyl]-4-phenyl-1H-imidazol-5-yl}-1H-pyrrol-1-yl)acetamide
(4-{[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}quinazolin-2-yl)methanol
1-[(3-methoxyphenyl)methyl]-N-[2-(naphthalen-1-yl)propan-2-yl]-6-oxopiperidine-3-carboxamide
5-{2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-propylpiperidin-4-yl)acetamide
4-{3-[(diethylamino)methyl]-4-methoxyphenyl}-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
N-methyl-N-(1-methylpiperidin-4-yl)-2-[(thiophen-2-ylmethyl)amino]benzamide
2-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}-N-(prop-2-en-1-yl)aniline
methyl[(1-methyl-1H-imidazol-5-yl)methyl]{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-{5-[2-(morpholin-4-yl)ethyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
1'-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-{[1-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}benzonitrile
3-(azocan-1-yl)-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]propanamide
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-{[4-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carbonyl)morpholine
2,3-dimethyl-7-[(1R,2S)-2-propylcyclopropanecarbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(2-methylpropanesulfonyl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]acetamide
N-{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
5-(oxolane-3-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S)-2-acetamido-3-(1H-imidazol-4-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
1-tert-butyl-4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
4-(4-ethylphenyl)-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-oxo-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-dihydroquinoline-4-carboxamide
2-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
(5S,9aS,9bS)-2-methyl-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
(2S,4S)-N-ethyl-4-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-amido}-1-propylpyrrolidine-2-carboxamide
2-amino-6-[4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-1-yl]-3,4-dihydropyrimidin-4-one
3-cyclopropyl-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-1H-pyrazole-5-carboxamide
4-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
4-{3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
3-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}urea
N-[3-methyl-1-(pyridin-3-yl)butyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
methyl N-(1-oxo-1-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}propan-2-yl)carbamate
3-[2-(2-methoxyethoxy)phenyl]-1-methyl-1-{[3-(methylsulfanyl)phenyl]methyl}urea