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3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide
N-[4-({7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenyl]acetamide
2-({2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-hydroxy-1-(2-methoxyethyl)-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
4-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
[(3R,4S)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-amino-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]benzonitrile
(3S,4R)-4-(hydroxymethyl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-3-ol
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(3S,4S)-1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
10-methoxy-5-(1H-1,2,3-triazole-5-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
7-(oxan-4-yl)-2-{2-[(trifluoromethyl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-(3,4-dimethylphenoxy)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]propan-1-ol
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
1-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-cyclobutanecarbonyl-4-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]piperidine
2-(1,2-benzoxazol-3-yl)-1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-2-ol
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amine
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
ethyl 1-[(2S)-2-acetamido-4-(methylsulfanyl)butanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
4-methyl-2-(pyridin-3-yl)-5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]pyrimidine
2-(2H-1,3-benzodioxol-5-yl)-1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]ethan-1-one
6-[4-(2,2,2-trifluoroethyl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
4-ethyl-3-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-{2-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-ethyl-5-(2-fluorophenoxymethyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
7-(5-chloropyridin-2-yl)-4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1λ6-thiomorpholine-1,1-dione
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-methylfuran-3-carboxamide
(4aS,7aR)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(1-methoxybutan-2-yl)-5-methyl-1H-pyrazole-4-carboxamide
2-{[2-(oxolan-3-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-1-(2-methylquinolin-6-yl)urea
2-cyclooctyl-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
2,4-dimethyl-N-{2-[7-(2-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
5-{3-[1-(pyrrolidin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-[3-(4-methylpiperazin-1-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(1H-imidazol-2-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
(3S,4S)-4-cyclopropyl-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
3-[benzyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]-2-methylpropan-1-ol