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1-(1-benzofuran-5-ylmethyl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
3-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1,3-diazepane-2,4-dione
1-[3-(5-methylfuran-2-yl)butyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
methyl (2S)-1-[9-methoxy-7-oxo-3-(3-phenylpropanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
N-methyl-3-(2-methylquinolin-5-yl)benzamide
N-[(2R,3R)-1'-(cyclopent-1-ene-1-carbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-({9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)phenol
N-(3-chloro-4-methoxyphenyl)-2-(3-methoxypropyl)piperidine-1-carboxamide
1-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
5-{2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-phenylpiperazine
ethyl 1-[(3-hydroxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-{2-[1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
2-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
methyl 5-[(2,5-dimethoxyphenyl)carbamoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
1'-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-[(3S,4S)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)pyrrolidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-(propan-2-yl)-3-propyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
1-methyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
1-(4-benzylpiperidin-1-yl)-3-[1-(furan-3-carbonyl)piperidin-4-yl]propan-1-one
N-[2-(5-cyclopentyl-4-phenyl-1H-imidazol-1-yl)ethyl]methanesulfonamide
2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-3-methyl-1H-indole
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}propanamide
2-(2,3-dimethylphenyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
1-[(3-methoxyphenyl)methyl]-4-(1-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
1-[2-methoxy-5-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-hydroxyphenyl)ethan-1-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(furan-2-carbonyl)piperidine-3-carboxylate
N-[(5-methylpyrazin-2-yl)methyl]-2-(morpholin-3-yl)acetamide
5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dimethylbenzene-1-sulfonamide
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(3-methoxyphenyl)ethan-1-one
5-benzamido-1-cyclopentyl-N-(3-hydroxy-2,2-dimethylpropyl)-1H-1,3-benzodiazole-7-carboxamide
methyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](pyrazin-2-ylmethyl)amine
methyl 3-{1-[2-(furan-2-yl)ethyl]-1H-imidazol-2-yl}benzoate
1-methyl-4-[(3E)-4-methylhex-3-en-1-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{1-[(3S,4R)-4-methoxyoxolan-3-yl]-4-phenyl-1H-imidazol-5-yl}-1-methyl-1H-1,3-benzodiazole
2-(2,5-dimethoxyphenyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetic acid
2-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)propan-2-ol
N-[(3R,4S)-1-cyclopentyl-4-propylpyrrolidin-3-yl]-2-(1,3-thiazol-4-yl)acetamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-[2-(3-chlorophenyl)acetyl]-4-propyl-1,4-diazepan-5-one
4-(2-butoxybenzoyl)-2-(trifluoromethyl)morpholine
2-(2-{4-[(ethylcarbamoyl)amino]-3-methoxyphenyl}-4-methylphenoxy)acetamide
4-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
1-[1'-(2-hydroxy-3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one