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3-(azepan-1-yl)-N-(2,5-dimethoxyphenyl)-3-oxopropanamide
1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butan-1-one
4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2-phenylmorpholine
N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-1H-1,3-benzodiazole-2-carboxamide
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(trimethyl-1H-imidazol-2-yl)methyl]pyrimidin-2-amine
{3-[(2,4-difluorophenyl)methyl]-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl}methanol
1-ethyl-4-{[methyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
[(3R,4R)-1-{[4-(2-aminoethyl)phenyl]methyl}-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethoxybenzamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]benzamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(1H-indol-2-ylmethyl)piperidine-4-carboxamide
2-(2-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
[2-(2-chlorophenoxy)ethyl](1-methoxypropan-2-yl)amine
N-[(2R,3R)-1'-(2,5-dimethylfuran-3-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-fluorobenzamide
N-(furan-2-ylmethyl)-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-methyl-1-[2-(piperazin-1-yl)ethyl]-N-(quinoxalin-6-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[2-(2-ethoxyphenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
1-(3-phenylpropyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
N-methyl-3-(5-methylthiophen-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
4-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
2-(methylsulfanyl)-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}benzoic acid
(5S)-5-[({[2-(5-methylfuran-2-yl)phenyl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-[3-(methylsulfanyl)phenyl]urea
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
3-methoxy-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)propanamide
N-(4-chloro-3-methylphenyl)-2-[(3S)-3-acetamidopyrrolidin-1-yl]acetamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-({7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
8-(2-cyclohexyl-1,3-benzoxazole-6-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-amido]cyclopentane-1-carboxylic acid
5-acetyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylthiophene-2-carboxamide
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-butyl-1-methyl-N-(pyridin-4-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
2-{3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}pyrazine
(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[(3-methoxyphenyl)methyl]piperidin-4-yl)methanol
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-fluoro-N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}propanamide
4-[3-(prop-2-en-1-yloxy)benzoyl]-7-(pyrrolidin-1-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-(6-methyl-2-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(dimethyl-1,2-oxazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(5-ethylpyrimidin-2-yl)-5-[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
5-{[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]methyl}pyrimidin-2-amine
ethyl 1-(oxan-4-yl)-4-(2-phenylethyl)piperidine-4-carboxylate
2-{4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperazin-1-yl}pyridine-3-carbonitrile
2-(carbamoylamino)-N-[(3R,4S)-4-cyclopropyl-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl]acetamide
N-cyclobutyl-1-cyclopentyl-6-oxopiperidine-3-carboxamide