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N4-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
N-(2-fluorophenyl)-3-[1-(4-methoxypyridine-2-carbonyl)piperidin-3-yl]propanamide
N-(1,4-dioxan-2-ylmethyl)-3-(1H-indol-3-yl)propanamide
{4-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}methanol
5-ethyl-2-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}pyridine
4-[2-(morpholin-4-yl)ethyl]-N-(1-propyl-1H-1,2,3-triazol-4-yl)piperazine-1-carboxamide
2-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
1-cyclopropyl-5-oxo-N-[2-(1,3-thiazol-4-yl)ethyl]pyrrolidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
7-methyl-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
methyl 2-{[(4-fluorophenyl)methyl]sulfamoyl}-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(3-methyl-1H-1,2,4-triazol-5-yl)ethan-1-one
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1-methylpiperazine-2-carboxylic acid
N-(1-{1-[4-(dimethylamino)benzoyl]piperidin-4-yl}-2-(2-methylphenyl)ethyl)-N-methyl-2-(1H-pyrazol-1-yl)acetamide
5-methyl-4-(1-methyl-1H-pyrazole-3-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2,3,6-trimethylphenoxy)acetamide
4-[2-(piperidine-1-carbonyl)phenoxy]-1-(1,3-thiazol-2-yl)piperidine
5-(dimethylamino)-2-{2-[4-(ethanesulfonyl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
2-(2-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-4-(pyrazin-2-yl)phenoxy)acetic acid
(cyclopropylmethyl)({[1-(morpholin-4-yl)cycloheptyl]methyl})amine
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-6-oxo-1,6-dihydropyridine-3-carboxamide
(3aR,6aR)-2-cyclopentyl-5-[3-(methylsulfanyl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{5-[1-(methoxymethyl)cyclobutanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
(4aR,7aS)-1-benzyl-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclobutyl-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
1-{2-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}piperidin-2-one
1-(carbamoylmethyl)-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]piperidine-4-carboxamide
3-[2-(piperazin-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
6-methoxy-3-{2-[3-methyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-indol-2-one
(3S,4R)-3-benzyl-1-(4-chloro-1H-pyrazole-3-carbonyl)-4-methylpiperidin-4-ol
2-chloro-6-fluoro-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-methylbenzamide
1-{1'-[5-(hydroxymethyl)furan-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-{[7-(2-cyclopentylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
2-(5-chloro-2-ethoxyphenyl)-1-(propan-2-yl)-1H-imidazole
(2-methoxyethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})propylamine
(2R,3R)-3-(1H-imidazol-1-yl)-1'-[(6-methylpyridin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(furan-2-ylmethyl)-N-methyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-N-[(5-methylfuran-2-yl)methyl]-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxylate
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[6-(4-methylphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
6-ethyl-2-methyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
1-[1-(4-methylpentyl)-7-oxoazepan-4-yl]-4-(piperidin-1-yl)piperidine-4-carboxamide
8-(5-chloropyridine-3-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-methyl-5-propylpyrimidin-4-amine
2-[1-(2-chloro-4-fluorobenzoyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
N-[2-(dimethylamino)ethyl]-4-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
5-methoxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]furan-2-carboxamide